SCHEMBL28037291

SCHEMBL28037291

C#CC[C@@H]([C@H](O)c1cc(F)ccc1F)N(C(=O)O)C(C)(C)C

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
RIPK1 Q13546 3/20 0.33
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
SLC6A4 P31645 4/20 0.31
SLC6A2 P23975 3/20 0.31
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31
APH1B Q8WW43 1/20 0.31
NCSTN Q92542 1/20 0.31
APH1A Q96BI3 1/20 0.31
PSENEN Q9NZ42 1/20 0.31
KCNQ4 P56696 1/20 0.30
KCNQ5 Q9NR82 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28037292 1.00 CES2 (0.36) CES2CES1RIPK1MAOAMAOB
SCHEMBL28062336 0.87 MAOA (0.32) MAOAMAOB
SCHEMBL28062335 0.87 MAOA (0.32) MAOAMAOB
SCHEMBL17102154 0.75 CES2 (0.40) CES2CES1RIPK1
SCHEMBL15524008 0.72 CES2 (0.40) CES2CES1MAOAMAOBPSEN1
SCHEMBL15524498 0.72 CES2 (0.40) CES2CES1MAOAMAOBPSEN1
SCHEMBL15524496 0.72 CES2 (0.40) CES2CES1MAOAMAOBPSEN1
SCHEMBL19712089 0.72 CES2 (0.40) CES2CES1MAOAMAOBPSEN1
SCHEMBL15524009 0.72 CES2 (0.40) CES2CES1MAOAMAOBPSEN1
SCHEMBL17380662 0.70 TRPA1 (0.41) CES2CES1KCNQ4KCNQ5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105531277-A Pyrrolo-imidazole ring derivatives and their use in medicine SICHUAN HAISCO PHARMACEUTICAL CO LTD 2016-04-27 CN disclosed
CN-105518008-A Amino pyranoid ring derivative and composition and use thereof SICHUAN HAISCO PHARMACEUTICAL CO LTD 2016-04-20 CN disclosed
CN-105294694-A Amino hexatomic ring derivative and application thereof to medicine SICHUAN HAISCO PHARMACEUTICAL CO LTD 2016-02-03 CN disclosed
CN-105085530-A Fused tricyclic substituted amino six-membered ring derivative and application thereof in medicine SICHUAN HAISCO PHARMACEUTICAL CO LTD 2015-11-25 CN disclosed
CN-105037367-A Amino six-membered ring derivative and application thereof in medicines SICHUAN HAISCO PHARMACEUTICAL CO LTD 2015-11-11 CN disclosed