SCHEMBL28037490

SCHEMBL28037490

COc1cccc(C(=O)NCCN(C)C)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.65
ALDH1A1 P00352 3/20 0.61
GAA P10253 2/20 0.61
MAPT P10636 1/20 0.61
L3MBTL1 Q9Y468 2/20 0.60
KMT2A Q03164 2/20 0.60
MEN1 O00255 1/20 0.60
TDP1 Q9NUW8 1/20 0.60
SMN1; SMN2 Q16637 4/20 0.58
HPGD P15428 3/20 0.58
MMP13 P45452 1/20 0.58
NPC1 O15118 4/20 0.57
RAB9A P51151 4/20 0.57
CYP2C9 P11712 1/20 0.57
CYP2C19 P33261 1/20 0.57
LMNA P02545 1/20 0.57
CYP2D6 P10635 1/20 0.56
TP53 P04637 1/20 0.56
HTT P42858 1/20 0.56
HSD17B10 Q99714 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3657784 0.92 SIGMAR1 (0.72) SIGMAR1ALDH1A1GAAMAPTL3MBTL1
SCHEMBL1499551 0.90 PDE4B (0.56) SIGMAR1ALDH1A1GAAMAPTL3MBTL1
SCHEMBL27792610 0.85 ALDH1A1 (0.51) SIGMAR1ALDH1A1GAAMAPTL3MBTL1
SCHEMBL8783271 0.84 SIGMAR1 (0.57) SIGMAR1ALDH1A1GAAMAPTL3MBTL1
SCHEMBL27951641 0.84 ALDH1A1 (0.65) SIGMAR1ALDH1A1GAAMAPTL3MBTL1
SCHEMBL30098865 0.84 ALDH1A1 (0.73) ALDH1A1GAAMAPTL3MBTL1KMT2A
SCHEMBL9491894 0.84 GAA (0.73) SIGMAR1ALDH1A1GAAMAPTL3MBTL1
SCHEMBL11756934 0.84 GAA (0.73) SIGMAR1ALDH1A1GAAMAPTL3MBTL1
SCHEMBL6361446 0.84 GAA (0.73) ALDH1A1GAAMAPTL3MBTL1KMT2A
SCHEMBL1499442 0.83 MTNR1B (0.54) ALDH1A1KMT2ASMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105073725-A Pyrazolyl-ureas as kinase inhibitors RESPIVERT LTD 2015-11-18 CN disclosed