SCHEMBL28037510

SCHEMBL28037510

O=CC1CN=C(c2ccccc2)c2cc(Cl)ccc2N1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 2/20 0.56
CNR1 P21554 1/20 0.56
NTSR1 P30989 1/20 0.56
PDE4D Q08499 1/20 0.56
CHRM1 P11229 7/20 0.53
ALDH1A1 P00352 1/20 0.53
PKM P14618 1/20 0.53
HTT P42858 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
ALB P02768 2/20 0.48
MEN1 O00255 1/20 0.48
LMNA P02545 1/20 0.48
KMT2A Q03164 1/20 0.48
CCKBR P32239 2/20 0.46
CCNE2 O96020 1/20 0.43
CCNE1 P24864 1/20 0.43
CDK2 P24941 1/20 0.43
GABRP O00591 1/20 0.43
GABRD O14764 1/20 0.43
CACNA1F O60840 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28333618 0.87 CHRM1 (0.56) OPRK1CNR1NTSR1PDE4DCHRM1
SCHEMBL28536668 0.86 GABRA1 (0.57) OPRK1CNR1NTSR1PDE4DCHRM1
SCHEMBL27689076 0.85 OPRK1 (0.39) OPRK1CNR1NTSR1PDE4DCHRM1
SCHEMBL27533159 0.84 LMNA (0.59) CHRM1LMNACCNE2CCNE1CDK2
SCHEMBL27390735 0.84 GABRA1 (0.50) OPRK1CNR1NTSR1PDE4DCHRM1
SCHEMBL27304815 0.82 CNR1 (0.38) OPRK1CNR1NTSR1PDE4DCHRM1
SCHEMBL28150316 0.81 CNR1 (0.39) OPRK1CNR1NTSR1PDE4DCHRM1
SCHEMBL27717603 0.81 LMNA (0.60) OPRK1PDE4DCHRM1ALDH1A1MEN1
SCHEMBL27663056 0.79 LMNA (0.47) OPRK1CNR1NTSR1PDE4DCHRM1
SCHEMBL10672472 0.77 CHRM1 (0.53) OPRK1CNR1NTSR1PDE4DCHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118290353-A Preparation method of stable isotope labeled diazepam 司法鉴定科学研究院 2024-07-05 CN claimed
CN-110579546-B Method for measuring alprazolam tablet related substances by high performance liquid chromatography 北京悦康科创医药科技股份有限公司 2022-05-03 CN claimed
CN-118290353-A Preparation method of stable isotope labeled diazepam 司法鉴定科学研究院 2024-07-05 CN disclosed
CN-118290353-A Preparation method of stable isotope labeled diazepam 司法鉴定科学研究院 2024-07-05 CN disclosed
CN-112500359-B Preparation method of lorazepam intermediate 华中药业股份有限公司 2022-06-03 CN disclosed
CN-110579546-B Method for measuring alprazolam tablet related substances by high performance liquid chromatography 北京悦康科创医药科技股份有限公司 2022-05-03 CN disclosed
CN-112500359-A Preparation method of lorazepam intermediate 华中药业股份有限公司 2021-03-16 CN disclosed
CN-110579546-A Method for measuring alprazolam tablet related substances by high performance liquid chromatography 北京悦康科创医药科技股份有限公司 2019-12-17 CN disclosed
CN-104961692-A Improved preparation method of 7-chlorin-5-phenyl-1,3-dihydro-2H-1,4-benzodiazepine-2-keto-4-oxide HUAZHONG PHARMACEUTICAL CO LTD 2015-10-07 CN disclosed