SCHEMBL28038544

SCHEMBL28038544

COc1nc(Cl)c2c(OC)c(OC)ccc2n1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.51
PDE3A Q14432 2/20 0.51
AMY1A P0DUB6 2/20 0.39
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 2/20 0.39
HPGD P15428 2/20 0.39
HSD17B10 Q99714 2/20 0.39
MAPK1 P28482 1/20 0.39
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
CYP1A1 P04798 2/20 0.37
CYP1B1 Q16678 2/20 0.37
MAT2A P31153 1/20 0.37
CYP19A1 P11511 1/20 0.36
HTT P42858 1/20 0.35
NQO2 P16083 1/20 0.34
CYP1A2 P05177 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2948476 0.85 PDE3B (0.53) PDE3BPDE3AAMY1AALDH1A1KDM4E
SCHEMBL10759980 0.81 PDE3B (0.49) PDE3BPDE3AAMY1AALDH1A1KDM4E
SCHEMBL27671629 0.78 ALDH1A1 (0.51) AMY1AALDH1A1KDM4EHPGDMAPT
SCHEMBL8807809 0.75 EGFR (0.48) PDE3BPDE3AAMY1AALDH1A1KDM4E
SCHEMBL4738100 0.72 PDE3A (0.50) PDE3BPDE3AAMY1AALDH1A1HPGD
SCHEMBL8374763 0.72 PDE3B (0.44) PDE3BPDE3AALDH1A1KDM4EHPGD
SCHEMBL27248807 0.69 PDE3B (0.40) PDE3BPDE3AAMY1AALDH1A1KDM4E
SCHEMBL27248563 0.69 ALDH1A1 (0.37) PDE3BPDE3AALDH1A1KDM4EHSD17B10
SCHEMBL275910 0.69 CYP1A2 (0.48) ALDH1A1GAAMAPTMAT2AHTT
SCHEMBL14353311 0.68 DCPS (0.63) PDE3BPDE3AALDH1A1HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105037279-B 4 N substituted quinazolines analog derivatives of the structure containing pentadienone and preparation and application 贵州大学 2017-11-03 CN disclosed
CN-105037279-A 4-N substituted quinazoline derivants adopting pentadienone structure and preparation and application of 4-N substituted quinazoline derivants UNIV GUIZHOU 2015-11-11 CN disclosed