SCHEMBL28039715

SCHEMBL28039715

OC1(c2ccccc2)C=CC=N1

nearest known ligand 0.32

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
OPRK1 P41145 1/20 0.31
OPRL1 P41146 1/20 0.31
P2RX1 P51575 1/20 0.30
P2RX3 P56373 1/20 0.30
P2RX4 Q99571 1/20 0.30
P2RX7 Q99572 1/20 0.30
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methane SCHEMBL28848706 0.98 OPRM1 (0.30) OPRM1OPRD1OPRK1OPRL1
SCHEMBL28833868 0.92
SCHEMBL27809189 0.73 ALDH1A1 (0.31)
SCHEMBL9877949 0.71 PNMT (0.35)
SCHEMBL27972084 0.71 ALDH1A1 (0.30)
SCHEMBL9034778 0.70 ALDH1A1 (0.38) OPRM1OPRK1OPRL1MEN1KMT2A
SCHEMBL1330599 0.69 AKR1C1 (0.37) KMT2A
SCHEMBL2164968 0.69 HTT (0.43) NPC1RAB9AKMT2A
SCHEMBL1067618 0.67 OPRL1 (0.33) OPRM1OPRD1OPRK1OPRL1P2RX1
SCHEMBL28917498 0.65 MAOB (0.31) OPRM1OPRK1OPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105008367-B It is used as the pyrrolo-triazine class compound of potassium channel inhibitors 百时美施贵宝公司 2017-08-29 CN disclosed
CN-105008367-A Pyrrolotriazines as potassium ion channel inhibitors BRISTOL MYERS SQUIBB CO 2015-10-28 CN disclosed