SCHEMBL28040113

SCHEMBL28040113

C=Cc1ccc(-c2ccccc2)n1Cc1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
HPGDS O60760 1/20 0.41
IDO1 P14902 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
CNR1 P21554 1/20 0.40
ALDH1A1 P00352 8/20 0.39
HPGD P15428 3/20 0.39
HSD17B10 Q99714 2/20 0.39
KMT2A Q03164 1/20 0.39
CYP19A1 P11511 2/20 0.39
LMNA P02545 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
RAB9A P51151 2/20 0.39
RECQL P46063 1/20 0.39
PDE6D O43924 1/20 0.38
ALDH2 P05091 1/20 0.38
ALDH3A1 P30838 1/20 0.38
NPSR1 Q6W5P4 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9664824 0.81 CYP19A1 (0.50) KDM4EL3MBTL1HPGDSIDO1CYP11B1
SCHEMBL20937641 0.81 KDM4E (0.46) KDM4EL3MBTL1ALDH1A1HPGDHSD17B10
SCHEMBL2263350 0.71 CNR1 (0.48) KDM4EL3MBTL1HPGDSCNR1ALDH1A1
SCHEMBL2825301 0.69 TSHR (0.48) KDM4EHPGDSIDO1CYP11B1CYP11B2
SCHEMBL4428277 0.69 NOTUM (0.48) KDM4EL3MBTL1CNR1ALDH1A1HPGD
SCHEMBL2260831 0.68 GSK3A (0.48) KDM4EHPGDSIDO1CYP11B1CYP11B2
SCHEMBL2261486 0.68 KDM4E (0.71) KDM4EL3MBTL1CNR1ALDH1A1HPGD
SCHEMBL20853006 0.68 CCR2 (0.54) KDM4EL3MBTL1ALDH1A1HPGDKMT2A
SCHEMBL28035380 0.66 HDAC8 (0.47) KDM4EL3MBTL1ALDH1A1SMN1; SMN2RAB9A
SCHEMBL10430575 0.64 KMT2A (0.49) KDM4ECNR1ALDH1A1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105008367-B It is used as the pyrrolo-triazine class compound of potassium channel inhibitors 百时美施贵宝公司 2017-08-29 CN disclosed
CN-105008367-A Pyrrolotriazines as potassium ion channel inhibitors BRISTOL MYERS SQUIBB CO 2015-10-28 CN disclosed