SCHEMBL28040274

SCHEMBL28040274

CC(C)(C)OC(=O)C(C(=O)C[N+](=O)[O-])C(N)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 1/20 0.38
ITGB7 P26010 1/20 0.38
FAAH O00519 1/20 0.36
ALDH1A1 P00352 3/20 0.36
CYP3A4 P08684 1/20 0.36
AAK1 Q2M2I8 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
GSR P00390 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
MAPT P10636 2/20 0.34
RECQL P46063 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
LTA4H P09960 1/20 0.34
CPA1 P15085 3/20 0.34
ATM Q13315 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28031607 0.82 CTSK (0.39) ALDH1A1AAK1CTSSCTSKKMT2A
SCHEMBL27875653 0.81 AAK1 (0.38) ITGA4ITGB7ALDH1A1AAK1CTSS
SCHEMBL27894672 0.81 AAK1 (0.38) ITGA4ITGB7ALDH1A1AAK1CTSS
SCHEMBL9832084 0.79 ALDH1A1 (0.41) ITGA4ITGB7ALDH1A1CYP3A4AAK1
SCHEMBL27665873 0.79 DPP4 (0.42) ALDH1A1AAK1CTSSCTSKMEN1
SCHEMBL4937584 0.79 DPP4 (0.42) ALDH1A1AAK1CTSSCTSKMEN1
SCHEMBL27564999 0.79 DPP4 (0.42) ALDH1A1AAK1CTSSCTSKMEN1
SCHEMBL8069348 0.79 ALDH1A1 (0.40) ITGA4ITGB7ALDH1A1CYP3A4AAK1
SCHEMBL28261977 0.78 ATM (0.44) ALDH1A1AAK1CTSSCTSKMEN1
SCHEMBL28837744 0.78 DPP4 (0.41) ALDH1A1CYP3A4AAK1CTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105085323-B Novel synthesis process of Darunavir intermediate 重庆圣华曦药业股份有限公司 2017-02-15 CN claimed
CN-105085323-A Novel synthesis process of Darunavir intermediate CHONGQING SHENGHUAXI PHARMA CO 2015-11-25 CN claimed
CN-105085323-B Novel synthesis process of Darunavir intermediate 重庆圣华曦药业股份有限公司 2017-02-15 CN disclosed
CN-105085323-A Novel synthesis process of Darunavir intermediate CHONGQING SHENGHUAXI PHARMA CO 2015-11-25 CN disclosed