SCHEMBL28031607

SCHEMBL28031607

CCC(=O)C(C(=O)OC(C)(C)C)C(N)c1ccccc1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.39
AAK1 Q2M2I8 1/20 0.39
CTSS P25774 1/20 0.39
CYP1A2 P05177 2/20 0.38
ALDH1A1 P00352 1/20 0.38
ATM Q13315 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
LTA4H P09960 1/20 0.37
CYP2D6 P10635 1/20 0.37
PKM P14618 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
DPP4 P27487 2/20 0.37
KMT2A Q03164 1/20 0.37
SLC7A5 Q01650 1/20 0.36
SYK P43405 1/20 0.36
MMP8 P22894 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27875653 0.87 AAK1 (0.38) CTSKAAK1CTSSCYP1A2ALDH1A1
SCHEMBL27894672 0.87 AAK1 (0.38) CTSKAAK1CTSSCYP1A2ALDH1A1
SCHEMBL27613183 0.85 MMP8 (0.41) CTSKCTSSL3MBTL1LTA4HCYP2D6
SCHEMBL9832084 0.85 ALDH1A1 (0.41) CTSKAAK1CTSSCYP1A2ALDH1A1
SCHEMBL4937584 0.84 DPP4 (0.42) CTSKAAK1CTSSCYP1A2ALDH1A1
SCHEMBL27564999 0.84 DPP4 (0.42) CTSKAAK1CTSSCYP1A2ALDH1A1
SCHEMBL27665873 0.84 DPP4 (0.42) CTSKAAK1CTSSCYP1A2ALDH1A1
SCHEMBL28837744 0.83 DPP4 (0.41) CTSKAAK1CTSSCYP1A2ALDH1A1
SCHEMBL28261977 0.83 ATM (0.44) CTSKAAK1CTSSCYP1A2ALDH1A1
SCHEMBL28040274 0.82 ITGA4 (0.38) CTSKAAK1CTSSALDH1A1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105017181-A Carfilzomib key intermediate and preparation method of its derivative UNIV NANJING NORMAL 2015-11-04 CN disclosed