SCHEMBL28040342

SCHEMBL28040342

FC(F)(F)c1ccnc(Sc2ccc(Br)cc2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 4/20 0.42
KDM4E B2RXH2 1/20 0.39
LRRK2 Q5S007 1/20 0.38
CHRNA7 P36544 1/20 0.36
HPGD P15428 2/20 0.35
ATM Q13315 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
HDAC3 O15379 1/20 0.35
NCOR1 O75376 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
ADRB1 P08588 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6250182 0.72 ADRB1 (0.40) SYKLRRK2HDAC3NCOR1HDAC4
SCHEMBL1184986 0.72 SYK (0.43) SYKKDM4ELRRK2HPGDATM
SCHEMBL29906009 0.72 SYK (0.43) SYKKDM4ELRRK2HPGDATM
SCHEMBL28135251 0.71 MEN1 (0.51) SYKKDM4EATMHDAC4ADRB1
SCHEMBL3903500 0.70 LRRK2 (0.40) LRRK2ATML3MBTL1HDAC3NCOR1
SCHEMBL1337601 0.69 ADRB1 (0.43) SYKADRB1LOXL2
SCHEMBL3903492 0.68 LRRK2 (0.37) SYKLRRK2HDAC3NCOR1HDAC4
SCHEMBL8345900 0.68 HDAC3 (0.42) SYKKDM4ELRRK2HDAC3NCOR1
SCHEMBL28040870 0.68 NOS3 (0.43) ATML3MBTL1ADRB1GRM5MEN1
SCHEMBL15390391 0.66 KMT2A (0.61) SYKHPGDL3MBTL1HDAC3NCOR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105085482-B Substituted diethylenediamine compound and its application method and purposes 广东东阳光药业有限公司 2018-08-10 CN disclosed
CN-105085482-A Substituted piperazine compound, and usage method and application thereof GUANGDONG HEC PHARMACEUTICAL 2015-11-25 CN disclosed