SCHEMBL28041367

SCHEMBL28041367

Cc1ccc2nc(N)c(-c3ccccc3)c(-c3ccccc3)c2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.50
ALDH1A1 P00352 4/20 0.50
MAPT P10636 4/20 0.50
LMNA P02545 3/20 0.50
L3MBTL1 Q9Y468 2/20 0.49
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
HSD17B10 Q99714 1/20 0.47
RECQL P46063 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
PSMB5 P28074 1/20 0.45
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44
MAPK1 P28482 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
DHODH Q02127 1/20 0.43
NQO2 P16083 1/20 0.43
CYP1A1 P04798 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP1B1 Q16678 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28041606 0.89 KDM4E (0.47) KDM4EALDH1A1MAPTLMNAL3MBTL1
SCHEMBL29660570 0.84 KDM4E (0.57) KDM4EALDH1A1MAPTLMNAL3MBTL1
SCHEMBL4596211 0.84 KDM4E (0.57) KDM4EALDH1A1MAPTLMNAL3MBTL1
SCHEMBL28041579 0.80 DHODH (0.49) KDM4EALDH1A1MAPTL3MBTL1MEN1
SCHEMBL28823862 0.80 FABP4 (0.54) KDM4EALDH1A1MAPTLMNARAB9A
SCHEMBL28361368 0.79 ESR1 (0.64) KDM4EALDH1A1MAPTLMNAL3MBTL1
SCHEMBL28197192 0.79 KDM4E (0.60) KDM4EALDH1A1MAPTLMNAL3MBTL1
SCHEMBL28041598 0.78 KDM4E (0.56) KDM4EALDH1A1MAPTLMNAL3MBTL1
SCHEMBL861205 0.77 CYP1A1 (0.50) KDM4EALDH1A1MAPTLMNAL3MBTL1
SCHEMBL27956647 0.77 ESR1 (0.70) KDM4EALDH1A1MAPTLMNAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104086485-B Prepare the method for poly-substituted quinoline type aromatic ring pyridine derivate TSINGHUA UNIVERSITY (CN) 2016-03-30 CN disclosed