SCHEMBL28041579

SCHEMBL28041579

Nc1nc2ccc(F)cc2c(-c2ccccc2)c1-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 4/20 0.49
KDM4E B2RXH2 3/20 0.47
HTT P42858 2/20 0.47
POLB P06746 2/20 0.47
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 1/20 0.47
KMT2A Q03164 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C19 P33261 2/20 0.46
HPGD P15428 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
ADORA2A P29274 2/20 0.44
MAPT P10636 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
MAPK1 P28482 1/20 0.44
CYP2C9 P11712 1/20 0.43
PIK3CD O00329 1/20 0.43
PIK3CA P42336 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28823862 0.80 FABP4 (0.54) KDM4EHTTALDH1A1HPGDADORA2A
SCHEMBL28041367 0.80 KDM4E (0.50) DHODHKDM4EMEN1ALDH1A1KMT2A
SCHEMBL28041598 0.78 KDM4E (0.56) KDM4EHTTPOLBALDH1A1KMT2A
SCHEMBL72673 0.77 KDM4E (0.47) DHODHKDM4EHTTPOLBMEN1
SCHEMBL28823807 0.76 NPC1 (0.46) DHODHKDM4EALDH1A1L3MBTL1CYP1A2
SCHEMBL789402 0.73 CYP1A2 (0.41) DHODHKDM4EHTTPOLBMEN1
SCHEMBL9971755 0.73 ACHE (0.46) DHODHKDM4EHTTPOLBMEN1
SCHEMBL840416 0.72 CLK1 (0.51) DHODHKDM4EHTTPOLBMEN1
SCHEMBL2720125 0.72 RORC (0.53) DHODHKDM4EHTTPOLBMEN1
SCHEMBL2717330 0.72 DHODH (0.51) DHODHKDM4EHTTPOLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104086485-B Prepare the method for poly-substituted quinoline type aromatic ring pyridine derivate TSINGHUA UNIVERSITY (CN) 2016-03-30 CN disclosed