SCHEMBL28041869

SCHEMBL28041869

CC(=O)Nc1cccc(C(N)COC(=O)NC(C)(C)C)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
RAB9A P51151 2/20 0.42
POLB P06746 1/20 0.41
NR4A1 P22736 1/20 0.41
HSD17B10 Q99714 2/20 0.40
CYP1A2 P05177 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ADRB2 P07550 1/20 0.40
ADRB1 P08588 1/20 0.40
ADRB3 P13945 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TACR1 P25103 1/20 0.39
TSHR P16473 1/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
SLC6A3 Q01959 2/20 0.39
KCNH2 Q12809 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28830732 0.81 PSEN1 (0.44) ALDH1A1TSHRSLC6A2SLC6A4SLC6A3
SCHEMBL28076445 0.81 ALDH1A1 (0.40) ALDH1A1RAB9ALMNAAAK1
SCHEMBL27770762 0.81 MAPT (0.46) CYP1A2L3MBTL1ADRB2ADRB1ADRB3
SCHEMBL28136985 0.77 SLC6A2 (0.41) CYP1A2MEN1KMT2ATSHRCYP3A4
SCHEMBL4705983 0.76 ALDH1A1 (0.54) ALDH1A1RAB9APOLBNR4A1HSD17B10
SCHEMBL28041868 0.76 CA1 (0.45) ALDH1A1RAB9APOLBNR4A1HSD17B10
SCHEMBL28094567 0.75 DPP4 (0.39) ALDH1A1POLBSLC6A2SLC6A3MAPT
SCHEMBL18599484 0.75 ALDH1A1 (0.49) ALDH1A1RAB9APOLBNR4A1HSD17B10
SCHEMBL4598418 0.74 MEN1 (0.48) ALDH1A1RAB9APOLBNR4A1HSD17B10
SCHEMBL4598417 0.74 MEN1 (0.48) ALDH1A1RAB9APOLBNR4A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104981470-A Amino-substituted imidazo[1,2-a]pyridinecarboxamides and their use Bayer Pharma AG 2015-10-14 CN disclosed