SCHEMBL28042941

SCHEMBL28042941

C[C](C)CN1CC=C(c2c(Cl)cc(N)cc2Cl)CC1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.38
LMNA P02545 3/20 0.38
MAPT P10636 3/20 0.37
HTR6 P50406 5/20 0.37
SIGMAR1 Q99720 4/20 0.34
SUV39H2 Q9H5I1 1/20 0.33
GAA P10253 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
CCNT1 O60563 1/20 0.32
CDK9 P50750 1/20 0.32
DRD2 P14416 2/20 0.32
DRD3 P35462 2/20 0.32
DRD4 P21917 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27979569 0.77 DRD4 (0.47) KDM4ELMNAMAPTSIGMAR1GAA
SCHEMBL28096230 0.74 SIGMAR1 (0.57) KDM4ELMNAMAPTSIGMAR1DRD2
SCHEMBL23277150 0.73 KDM4E (0.49) KDM4ELMNAMAPTSIGMAR1DRD2
SCHEMBL27831844 0.73 KDM4E (0.41) KDM4ELMNAMAPTSIGMAR1SUV39H2
SCHEMBL27712204 0.70 KDM4E (0.43) KDM4ELMNAMAPTHTR6SIGMAR1
SCHEMBL16013186 0.70 PDK4 (0.52) HTR6
SCHEMBL27801629 0.70 KDM4E (0.56) KDM4ELMNAMAPTSIGMAR1GAA
SCHEMBL27979395 0.69 MEN1 (0.42) KDM4EMAPTSIGMAR1MEN1KMT2A
SCHEMBL27914131 0.68 SIGMAR1 (0.57) MAPTSIGMAR1MEN1KMT2ADRD2
SCHEMBL28108120 0.68 QDPR (0.51) KDM4EMAPTSIGMAR1SUV39H2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105051033-B Antiviral compound 豪夫迈·罗氏有限公司 2018-02-16 CN disclosed
CN-105051033-A Antiviral compounds HOFFMANN LA ROCHE 2015-11-11 CN disclosed