SCHEMBL28042985

SCHEMBL28042985

COC(=O)c1ccccc1OCBr

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 3/20 0.56
HTT P42858 2/20 0.54
HSP90AA1 P07900 2/20 0.54
MAPT P10636 2/20 0.54
NPSR1 Q6W5P4 1/20 0.54
KMT2A Q03164 3/20 0.53
ALDH1A1 P00352 4/20 0.52
TSHR P16473 2/20 0.52
KDM4E B2RXH2 1/20 0.52
LMNA P02545 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.51
MEN1 O00255 2/20 0.51
GAA P10253 1/20 0.51
CYP1A2 P05177 1/20 0.50
CYP2C9 P11712 1/20 0.50
HPGD P15428 1/20 0.50
CYP2C19 P33261 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
CFTR P13569 1/20 0.50
HSD17B10 Q99714 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2389931 0.86 HSP90AA1 (0.58) SLC6A3HTTHSP90AA1MAPTNPSR1
SCHEMBL6043498 0.85 MAPT (0.60) SLC6A3HTTHSP90AA1MAPTNPSR1
SCHEMBL1989129 0.84 HCRTR1 (0.65) SLC6A3HTTHSP90AA1MAPTNPSR1
SCHEMBL28136228 0.84 SLC6A3 (0.57) SLC6A3HTTHSP90AA1MAPTNPSR1
SCHEMBL30553984 0.84 HCRTR1 (0.65) SLC6A3HTTHSP90AA1MAPTNPSR1
SCHEMBL4385291 0.84 SLC6A3 (0.57) SLC6A3HTTHSP90AA1MAPTNPSR1
SCHEMBL16674272 0.83 TSHR (0.65) HTTMAPTKMT2AALDH1A1TSHR
SCHEMBL8399356 0.82 ALDH1A1 (0.59) SLC6A3HTTHSP90AA1MAPTNPSR1
SCHEMBL2005183 0.82 SLC6A3 (0.56) SLC6A3HTTHSP90AA1MAPTNPSR1
SCHEMBL2290004 0.82 SLC6A3 (0.56) SLC6A3HTTHSP90AA1MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105121427-B Pyridine radicals and condensed pyridine base triazolone derivative 武田药品工业株式会社 2018-04-10 CN disclosed
CN-105121427-A Pyridinyl and fused pyridinyl triazolone derivatives TAKEDA PHARMACEUTICAL 2015-12-02 CN disclosed
CN-105051048-A 1-hydroxy-benzoxaboroles as antiparasitic agents LILLY CO ELI 2015-11-11 CN disclosed