SCHEMBL28043073

SCHEMBL28043073

CNc1cc(-c2ccc(OC(F)(F)F)cc2)ccn1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SCN5A Q14524 3/20 0.46
ABL1 P00519 2/20 0.44
BCR P11274 1/20 0.44
SCN9A Q15858 1/20 0.44
KIF11 P52732 1/20 0.43
FDPS P14324 2/20 0.42
GSK3B P49841 3/20 0.42
GSK3A P49840 1/20 0.42
RAF1 P04049 1/20 0.42
EPHX2 P34913 1/20 0.42
SCN10A Q9Y5Y9 1/20 0.42
CHRNA7 P36544 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
WNT3A P56704 1/20 0.41
DYRK1A Q13627 1/20 0.41
GPR39 O43194 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23763117 0.82 RXRA (0.43) ABL1BCRRAF1EPHX2GPR39
SCHEMBL28043122 0.80 KIF11 (0.53) ABL1BCRKIF11GSK3BGSK3A
SCHEMBL25754727 0.80 DYRK1A (0.65) SCN5AABL1SCN9AKIF11SCN10A
SCHEMBL4325626 0.79 MAPK10 (0.68) ABL1BCRGSK3B
SCHEMBL28266489 0.77 GSK3B (0.64) ABL1GSK3BGSK3A
SCHEMBL6530522 0.77 MAPK10 (0.61)
Hydrochloric Acid SCHEMBL28074538 0.77 ABL1 (0.61) ABL1BCRADORA3
SCHEMBL1229896 0.76 SCN5A (0.49) SCN5AABL1BCRSCN9ADYRK1A
SCHEMBL13741332 0.76 SCN5A (0.49) SCN5AABL1BCRSCN9AKIF11
SCHEMBL25755093 0.76 SCN5A (0.46) SCN5AABL1SCN9AKIF11SCN10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143188-A Novel sulfonamide trpa1 receptor antagonists PHARMESTE S R L IN LIQUIDATION 2015-12-09 CN disclosed