SCHEMBL28043663

SCHEMBL28043663

CC(OC=O)c1c[nH]c2cc(N)ccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 4/20 0.38
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
HTR2A P28223 3/20 0.34
HTR2C P28335 2/20 0.34
HTR2B P41595 2/20 0.34
ASH1L Q9NR48 1/20 0.34
PARP1 P09874 1/20 0.33
FFAR1 O14842 1/20 0.33
GPR84 Q9NQS5 1/20 0.33
CLK1 P49759 1/20 0.33
CDK5 Q00535 1/20 0.33
CDK5R1 Q15078 1/20 0.33
CYP2A6 P11509 1/20 0.32
PLG P00747 1/20 0.31
PLAU P00749 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27648954 0.89 HTR2A (0.41) ALDH1A1HTR2AHTR2CHTR2BFFAR1
SCHEMBL27526971 0.84 NR4A2 (0.44) KDM4EALDH1A1MAPTHTR2AFFAR1
SCHEMBL27550865 0.83 NR4A2 (0.46) KDM4EALDH1A1MAPTHTR2AGPR84
SCHEMBL27528319 0.83 CYP2A6 (0.51) IMPDH2KDM4EALDH1A1MAPTCYP2A6
SCHEMBL27785494 0.83 HTR2C (0.40) KDM4EALDH1A1MAPTHTR2AHTR2C
SCHEMBL28658779 0.83 GPR84 (0.43) HTR2AHTR2CGPR84
SCHEMBL27552422 0.83 ALDH1A1 (0.35) KDM4EALDH1A1MAPTHTR2AHTR2C
SCHEMBL27792585 0.82 HTR2A (0.38) KDM4EALDH1A1MAPTHTR2AHTR2C
SCHEMBL28929780 0.82 ALDH1A1 (0.57) KDM4EALDH1A1MAPTHTR2AHTR2C
SCHEMBL28291597 0.81 PLG (0.42) IMPDH2KDM4EALDH1A1HTR2CASH1L

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105745192-A Substituted phenylalanine derivatives 拜耳制药股份公司 2016-07-06 CN disclosed
CN-105164122-A Substituted oxopyridine derivatives and their use in the treatment of cardiovascular disorders Bayer Pharma AG 2015-12-16 CN disclosed
CN-101790313-A Compound (I) SMITHKLINE BEECHAM CORP 2010-07-28 CN disclosed