SCHEMBL28043672

SCHEMBL28043672

OB(OBr)c1cccc(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.40
ORAI1 Q96D31 1/20 0.36
ORAI2 Q96SN7 1/20 0.36
ORAI3 Q9BRQ5 1/20 0.36
TRPV6 Q9H1D0 1/20 0.36
WDR5 P61964 1/20 0.36
ALDH1A1 P00352 2/20 0.35
ENPP2 Q13822 3/20 0.35
PARP1 P09874 1/20 0.34
HTR3E A5X5Y0 2/20 0.33
HTR3B O95264 2/20 0.33
HTR3A P46098 2/20 0.33
HTR3D Q70Z44 2/20 0.33
HTR3C Q8WXA8 2/20 0.33
CYP3A4 P08684 2/20 0.33
IDO1 P14902 2/20 0.33
AGXT P21549 2/20 0.33
ALOX5 P09917 1/20 0.33
SLC22A2 O15244 1/20 0.33
SLC22A1 O15245 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4437860 0.80 CYP3A4 (0.41) TSHRORAI1ORAI2ORAI3TRPV6
SCHEMBL19820142 0.80 ENPP2 (0.41) TSHRORAI1ORAI2ORAI3TRPV6
SCHEMBL7461964 0.80 TSHR (0.40) TSHRORAI1ORAI2ORAI3TRPV6
SCHEMBL31492054 0.77 TSHR (0.38) TSHRORAI1ORAI2ORAI3TRPV6
SCHEMBL11815 0.76 ENPP2 (0.56) TSHRORAI1ORAI2ORAI3TRPV6
SCHEMBL1138514 0.76 ORAI1 (0.54) TSHRORAI1ORAI2ORAI3TRPV6
SCHEMBL28878253 0.76 ACHE (0.42) ALDH1A1ENPP2PARP1HTR3EHTR3B
SCHEMBL4832666 0.74 CYP2D6 (0.36) TSHRORAI1ORAI2ORAI3TRPV6
SCHEMBL150115 0.73 TRPV6 (0.50) TSHRORAI1ORAI2ORAI3TRPV6
SCHEMBL28329900 0.73 ENPP2 (0.67) TSHRALDH1A1ENPP2PARP1HTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108409773-A Compound and its application containing triazine group and a kind of organic electroluminescence device 北京绿人科技有限责任公司 2018-08-17 CN disclosed
CN-108164513-A Substituted oxo pyridine derivative and its purposes in terms of cardiovascular disorder is treated 拜耳制药股份公司 2018-06-15 CN disclosed
CN-105164122-B Substituted oxopyridine derivatives and their use in the treatment of cardiovascular disorders 拜耳制药股份公司 2018-02-02 CN disclosed
CN-105164122-A Substituted oxopyridine derivatives and their use in the treatment of cardiovascular disorders Bayer Pharma AG 2015-12-16 CN disclosed