SCHEMBL28044065

SCHEMBL28044065

CC(C)(C)C(=O)ONc1ccccc1N

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 11/20 0.42
HDAC3 O15379 8/20 0.42
HDAC2 Q92769 8/20 0.42
MAPK1 P28482 1/20 0.42
HDAC10 Q969S8 4/20 0.42
HDAC6 Q9UBN7 4/20 0.42
HDAC4 P56524 3/20 0.42
HDAC7 Q8WUI4 3/20 0.42
HDAC11 Q96DB2 3/20 0.42
HDAC8 Q9BY41 3/20 0.42
HDAC9 Q9UKV0 3/20 0.42
HDAC5 Q9UQL6 3/20 0.42
ALDH1A1 P00352 1/20 0.41
CFTR P13569 1/20 0.41
HSD17B10 Q99714 1/20 0.41
NCOR2 Q9Y618 3/20 0.40
PTGS1 P23219 2/20 0.40
MAPK13 O15264 2/20 0.38
MAPK12 P53778 2/20 0.38
MAPK11 Q15759 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25502829 0.80 HDAC1 (0.46) HDAC1HDAC3HDAC2MAPK1HDAC10
SCHEMBL28090478 0.79 PDK1 (0.46) ALDH1A1NPC1RAB9AELANECETP
SCHEMBL28090565 0.79 LMNA (0.49) MAPK1ALDH1A1NPC1RAB9ALMNA
SCHEMBL28832949 0.79 PDK1 (0.51) ALDH1A1NPC1RAB9ALMNA
SCHEMBL28018573 0.78 KDM4E (0.52) ALDH1A1HSD17B10LMNA
SCHEMBL28339992 0.78 HDAC1 (0.44) HDAC1HDAC3HDAC2ALDH1A1NCOR2
SCHEMBL28876956 0.77 POLB (0.49) MAPK1ALDH1A1NPC1RAB9ALMNA
SCHEMBL28148996 0.74 ALDH1A1 (0.45) ALDH1A1HSD17B10NPC1RAB9AELANE
SCHEMBL31285956 0.73 HDAC3 (0.41) HDAC1HDAC3HDAC2MAPK1HDAC10
SCHEMBL2733296 0.73 CETP (0.61) HDAC1HDAC3HDAC2MAPK1HDAC10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103864792-B Heterocyclic nitrogen compound acting as tyrosine kinase inhibitor 山东亨利医药科技有限责任公司 2017-01-18 CN disclosed
CN-105367503-A HETEROARYL COMPOUNDS AND USES THEREOF AVILA THERAPEUTICS INC 2016-03-02 CN disclosed
CN-105188371-A Erk inhibitors and uses thereof CELGENE AVILOMICS RES INC 2015-12-23 CN disclosed
CN-101902911-B Heteroaryl compounds and uses thereof AVILA THERAPEUTICS, INC. (US) 2015-12-16 CN disclosed
CN-105120860-A Histone deacetylase inhibitors BIOMARIN PHARM INC 2015-12-02 CN disclosed