SCHEMBL28044112

SCHEMBL28044112

CC(OC=O)c1c[nH]c2cccc(OCC3CC3)c12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 1/20 0.34
PDE4A P27815 2/20 0.34
PDE4B Q07343 2/20 0.34
PDE4C Q08493 2/20 0.34
PDE4D Q08499 2/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HTR2A P28223 5/20 0.33
HPGD P15428 1/20 0.33
PDE5A O76074 1/20 0.33
BRD4 O60885 1/20 0.33
TP53 P04637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
ALOX15 P16050 1/20 0.32
ADRA1D P25100 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27891882 0.81 HTR2A (0.37) PDE4APDE4BPDE4CPDE4DMEN1
SCHEMBL27472077 0.81 HTR2A (0.51) MEN1KMT2AMAPTKDM4EALDH1A1
SCHEMBL28678155 0.80 HTR2A (0.45) MEN1KMT2AMAPTHTR2AHTR2C
SCHEMBL27908791 0.79 HTR2A (0.35) MEN1KMT2AMAPTKDM4EALDH1A1
SCHEMBL27369292 0.75 GPR84 (0.44) MEN1KMT2AMAPTKDM4EALDH1A1
SCHEMBL27524231 0.74 NR4A2 (0.46) PDE4DHTR2AHTR2CHTR2B
SCHEMBL27771264 0.74 HTR2A (0.44) MEN1KMT2AMAPTKDM4EALDH1A1
SCHEMBL27906752 0.74 FFAR1 (0.43) HTR2AHTR2CHTR2B
SCHEMBL27965809 0.74 CYP2A6 (0.35) HTR2AHTR2CHTR2B
SCHEMBL27580249 0.74 MEN1 (0.36) MEN1KMT2AMAPTKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105164130-A Dihydro-pyrrolopyridone bromodomain inhibitors ABBVIE INC 2015-12-16 CN disclosed