SCHEMBL28044331

SCHEMBL28044331

NN(Cc1ccc(O)cc1)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.53
ESR1 P03372 5/20 0.49
ALDH1A1 P00352 2/20 0.47
MEN1 O00255 1/20 0.47
HSP90AA1 P07900 1/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
KMT2A Q03164 1/20 0.47
LTB4R2 Q9NPC1 1/20 0.44
ESR2 Q92731 3/20 0.44
FNTA P49354 1/20 0.44
FNTB P49356 1/20 0.44
MTOR P42345 1/20 0.44
AOC3 Q16853 1/20 0.43
G6PC1 P35575 1/20 0.43
ABAT P80404 1/20 0.43
PDK1 Q15118 1/20 0.41
TAS2R14 Q9NYV8 1/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL544819 0.87 AOC3 (0.56) ESR1ALDH1A1MEN1HSP90AA1GAA
Hydrochloric Acid SCHEMBL4825334 0.85 AOC3 (0.54) ESR1ALDH1A1MEN1HSP90AA1GAA
SCHEMBL12016039 0.82 TP53 (0.50) ALDH1A1MEN1KMT2AAOC3TAS2R14
SCHEMBL9879437 0.82 SLC6A2 (0.47) CYP19A1MEN1KMT2AAOC3G6PC1
SCHEMBL8975208 0.81 TSHR (0.55) CYP19A1ESR1ALDH1A1MEN1HSP90AA1
SCHEMBL11874481 0.81 ESR1 (0.66) CYP19A1ESR1ALDH1A1MEN1HSP90AA1
Hydrochloric Acid SCHEMBL9518503 0.80 SLC6A2 (0.46) CYP19A1MEN1KMT2AAOC3G6PC1
SCHEMBL27493772 0.79 ALDH1A1 (0.50) ESR1ALDH1A1MEN1MAPTKMT2A
SCHEMBL4427377 0.78 CRHBP (0.57) CYP19A1ESR1ALDH1A1MEN1HSP90AA1
Hydrochloric Acid SCHEMBL28901400 0.77 CRHBP (0.58) CYP19A1ALDH1A1MEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105503747-A Novel quinazoline derivative LU1507 as well as preparation method and application thereof NANJING GENERAL HOSPITAL NANJING MILITARY AREA COMMAND PLA 2016-04-20 CN disclosed
CN-105481835-A Novel quinazoline derivative LU1508, and preparation method and application thereof NANJING GENERAL HOSPITAL NANJING MILITARY AREA COMMAND PLA 2016-04-13 CN disclosed