SCHEMBL28044533

SCHEMBL28044533

CN(CCN1CCCCC1)c1cc[c]c(NS(C)(=O)=O)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 4/20 0.47
SIGMAR1 Q99720 6/20 0.39
CCR2 P41597 1/20 0.39
LTA4H P09960 1/20 0.37
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
CYP2D6 P10635 2/20 0.34
MAPK1 P28482 2/20 0.34
GRIN2D O15399 1/20 0.34
GRIN3B O60391 1/20 0.34
TP53 P04637 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2A Q12879 1/20 0.34
GRIN2B Q13224 1/20 0.34
GRIN2C Q14957 1/20 0.34
GRIN3A Q8TCU5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28044536 0.77 HTR7 (0.33) HTR7
SCHEMBL28044453 0.77 HTR7 (0.33) HTR7
SCHEMBL592097 0.76 SIGMAR1 (0.42) HTR7SIGMAR1CCR2ESR1ESR2
SCHEMBL589726 0.76 NTSR1 (0.35) HTR7SIGMAR1CCR2HRH3CYP2D6
SCHEMBL592328 0.75 HTR7 (0.49) HTR7SIGMAR1CCR2ESR1ESR2
SCHEMBL1355876 0.67 SIGMAR1 (0.43) SIGMAR1HRH3CYP2D6MAPK1CYP3A4
SCHEMBL11144109 0.66 SIGMAR1 (0.57) HTR7SIGMAR1CCR2HRH3
SCHEMBL1355874 0.66 SIGMAR1 (0.41) SIGMAR1CYP2D6MAPK1TP53TSHR
SCHEMBL1355593 0.65 SIGMAR1 (0.41) SIGMAR1CYP2D6MAPK1CYP3A4
SCHEMBL28044442 0.65 NR3C1 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101594862-B Substituted indazole derivatives as kinase inhibitors NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2015-11-25 CN disclosed