SCHEMBL28045440

SCHEMBL28045440

COC(=O)c1ccc(NC(C)=O)s1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 2/20 0.64
GAA P10253 1/20 0.64
PKM P14618 1/20 0.64
HSD17B10 Q99714 1/20 0.64
L3MBTL1 Q9Y468 2/20 0.55
TDP1 Q9NUW8 1/20 0.55
NPSR1 Q6W5P4 2/20 0.51
LMNA P02545 2/20 0.51
PPARG P37231 1/20 0.51
NCOA2 Q15596 1/20 0.51
NCOA1 Q15788 1/20 0.51
NCOA3 Q9Y6Q9 1/20 0.51
MAPK1 P28482 2/20 0.49
CYP1A2 P05177 2/20 0.49
APOBEC3A P31941 1/20 0.49
APOBEC3G Q9HC16 1/20 0.49
HPGD P15428 4/20 0.46
TSHR P16473 2/20 0.46
ATM Q13315 1/20 0.46
P2RY1 P47900 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6735515 0.85 PKM (0.69) ALOX15GAAPKMHSD17B10L3MBTL1
SCHEMBL24142017 0.81 NPSR1 (0.55) ALOX15GAAPKMHSD17B10L3MBTL1
SCHEMBL1484339 0.80 L3MBTL1 (0.50) ALOX15GAAPKMHSD17B10L3MBTL1
SCHEMBL27877799 0.80 L3MBTL1 (0.50) ALOX15GAAPKMHSD17B10L3MBTL1
SCHEMBL70027 0.80 NPSR1 (0.67) HSD17B10L3MBTL1TDP1NPSR1LMNA
SCHEMBL24188302 0.79 HSD17B10 (0.67) ALOX15GAAPKMHSD17B10L3MBTL1
SCHEMBL380561 0.78 L3MBTL1 (0.49) ALOX15GAAPKMHSD17B10L3MBTL1
SCHEMBL12009447 0.78 GAA (0.64) ALOX15GAAPKMHSD17B10LMNA
SCHEMBL277203 0.76 LMNA (0.58) GAAL3MBTL1TDP1NPSR1LMNA
SCHEMBL10519422 0.75 GSK3B (0.61) ALOX15GAAPKMHSD17B10L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105111197-A Synthesis methods of raltitrexed SHANGHAI DINGYA PHARMACEUTICAL CHEMICALS CO LTD 2015-12-02 CN disclosed