SCHEMBL24142017

SCHEMBL24142017

CNc1ccc(C(=O)OC)s1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.55
LMNA P02545 1/20 0.55
PPARG P37231 1/20 0.55
NCOA2 Q15596 1/20 0.55
NCOA1 Q15788 1/20 0.55
NCOA3 Q9Y6Q9 1/20 0.55
L3MBTL1 Q9Y468 3/20 0.50
TDP1 Q9NUW8 2/20 0.50
HPGD P15428 4/20 0.49
TSHR P16473 3/20 0.49
ATM Q13315 2/20 0.49
MAPK1 P28482 2/20 0.49
KDM4E B2RXH2 3/20 0.40
ALDH1A1 P00352 2/20 0.40
POLB P06746 1/20 0.40
MRGPRX4 Q96LA9 1/20 0.39
P2RY1 P47900 1/20 0.39
OPRD1 P41143 1/20 0.38
PARP1 P09874 1/20 0.38
HSD17B10 Q99714 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28198399 0.83 DAO (0.54) HPGDKDM4EPOLBHSD17B10GAA
SCHEMBL70027 0.83 NPSR1 (0.67) NPSR1LMNAPPARGNCOA2NCOA1
SCHEMBL7257673 0.82 HDAC3 (0.55) NPSR1LMNAL3MBTL1HPGDTSHR
SCHEMBL28045440 0.81 ALOX15 (0.64) NPSR1LMNAPPARGNCOA2NCOA1
SCHEMBL23682740 0.79 LMNA (0.48) NPSR1LMNAL3MBTL1HPGDTSHR
SCHEMBL1235256 0.77 LMNA (0.60) NPSR1LMNAPPARGNCOA2NCOA1
SCHEMBL1303016 0.77 NPSR1 (0.60) NPSR1LMNAPPARGNCOA2NCOA1
SCHEMBL1587481 0.76 NPSR1 (0.55) NPSR1LMNAPPARGNCOA2NCOA1
SCHEMBL27861920 0.76 NPSR1 (0.46) NPSR1LMNAPPARGNCOA2NCOA1
SCHEMBL1484339 0.75 L3MBTL1 (0.50) NPSR1LMNAPPARGNCOA2NCOA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021262693-A1 METHOTREXATE ANALOGS AND METHODS OF USE THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2021-12-30 WO disclosed