SCHEMBL28045792

SCHEMBL28045792

O=COC(Cc1cccc(F)c1)Cc1c[nH]cn1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.36
MAOB P27338 2/20 0.36
KDM4E B2RXH2 1/20 0.35
SLC1A1 P43005 2/20 0.34
ROCK2 O75116 3/20 0.34
MAP3K7 O43318 1/20 0.33
TAB1 Q15750 1/20 0.33
PPARG P37231 1/20 0.33
PPARA Q07869 1/20 0.33
DAO P14920 1/20 0.33
CDC7 O00311 1/20 0.33
DBF4 Q9UBU7 1/20 0.33
AURKA O14965 1/20 0.33
DAPK3 O43293 1/20 0.33
JAK2 O60674 1/20 0.33
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33
PAK4 O96013 1/20 0.33
ABL1 P00519 1/20 0.33
LCK P06239 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28074772 0.85 CTSK (0.36) CYP1A2
SCHEMBL28260269 0.73 DAO (0.42) KDM4EDAOCDC7DBF4IDO1
SCHEMBL224676 0.72 TAAR1 (0.47) KDM4EDAOIDO1AGXT
SCHEMBL27617418 0.71 POLB (0.30)
SCHEMBL28763764 0.71 PCSK9 (0.38) KDM4EDAOIDO1
SCHEMBL28052170 0.68 KLKB1 (0.35)
SCHEMBL22503743 0.68 ROCK2 (0.45) SLC1A1ROCK2ROCK1
SCHEMBL15072037 0.68
SCHEMBL2104753 0.66 CYP19A1 (0.41) KDM4ESLC1A1PPARGPPARAIDO1
SCHEMBL28102233 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105121432-A Heterocyclic amides as kinase inhibitors GLAXOSMITHKLINE IP DEV LTD 2015-12-02 CN disclosed