SCHEMBL28074772

SCHEMBL28074772

O=COC(Cc1ccccc1)Cc1c[nH]cn1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSK P43235 6/20 0.36
CTSL P07711 2/20 0.34
CTSB P07858 2/20 0.34
EPHX1 P07099 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33
CTSH P09668 1/20 0.31
CPA1 P15085 1/20 0.31
LAP3 P28838 4/20 0.30
ANPEP P15144 1/20 0.30
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28045792 0.85 MAOA (0.36) CYP1A2
SCHEMBL18085416 0.80 EPHX1 (0.48) CTSKCTSLCTSBEPHX1MEN1
SCHEMBL28061404 0.79 EPHX1 (0.35) CTSKCTSLCTSBEPHX1MEN1
SCHEMBL28045730 0.77 CTSK (0.37) CTSKCTSLCTSBEPHX1MEN1
SCHEMBL28052170 0.76 KLKB1 (0.35)
SCHEMBL18065072 0.76
SCHEMBL15072037 0.73
SCHEMBL28113598 0.73 CTSK (0.34) CTSKCTSLCTSBEPHX1MEN1
SCHEMBL27698547 0.73 PNP (0.36) CTSKEPHX1CPA1CYP1A2
SCHEMBL31690300 0.72 CYP1A2 (0.61) CPA1ANPEPCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105829317-B Imidazopyrazines ketone derivatives 默克专利股份公司 2019-03-29 CN disclosed
CN-105829317-A Imidazopyrazinone derivatives 默克专利股份公司 2016-08-03 CN disclosed