SCHEMBL28045833

SCHEMBL28045833

O=C(O)c1cccc(B(O)OCl)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA6 P23280 1/20 0.46
CA9 Q16790 1/20 0.46
AKR1C3 P42330 1/20 0.44
TTR P02766 2/20 0.44
KMO O15229 3/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C9 P11712 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
RXRA P19793 1/20 0.42
RXRB P28702 1/20 0.42
UNG P13051 1/20 0.42
FOLH1 Q04609 1/20 0.41
DAO P14920 1/20 0.40
TSHR P16473 1/20 0.40
NAPRT Q6XQN6 1/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15999885 0.82 CA12 (0.46) CA12CA1CA2CA6CA9
SCHEMBL14970703 0.82 CA12 (0.46) CA12CA1CA2CA6CA9
SCHEMBL6684 0.79 TTR (0.59) CA12CA1CA2CA6CA9
SCHEMBL29380260 0.79 TTR (0.59) CA12CA1CA2CA6CA9
SCHEMBL8000294 0.78 TTR (0.44) CA12CA1CA2CA6CA9
SCHEMBL28159303 0.77 TTR (0.57) CA12CA1CA2CA6CA9
SCHEMBL29658033 0.74 MGLL (0.62) CA1CA2CA6KMO
SCHEMBL244920 0.74 TRPV6 (0.50) CA1CA2CA6CYP1A2HPGD
Benzene SCHEMBL28042387 0.74 TRPV6 (0.50) CA1CA2CA6CYP1A2HPGD
SCHEMBL17667917 0.73 ENPP2 (0.59) CA12CA1CA2CA6CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102724975-B IRE-1 alpha inhibitors MANNKIND CORP. (US) 2015-12-02 CN disclosed