SCHEMBL28045914

SCHEMBL28045914

Cc1c(-c2ccccc2)cn(C(N)=O)c1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 2/20 0.42
PARP1 P09874 1/20 0.39
MAPT P10636 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
PTGS1 P23219 1/20 0.37
PDCD1 Q15116 1/20 0.36
CD274 Q9NZQ7 1/20 0.36
LMNA P02545 1/20 0.35
MEN1 O00255 4/20 0.35
KMT2A Q03164 4/20 0.35
BRD4 O60885 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 3/20 0.35
GAA P10253 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11306415 0.76 ESR2 (0.40) MAPTSMN1; SMN2KDM4EALDH1A1CYP1A2
SCHEMBL27645536 0.74 BCAT2 (0.43) BCAT2PARP1MAPTNPC1LMNA
SCHEMBL7852845 0.71 ALDH1A1 (0.37) BCAT2MAPTNPC1RAB9ALMNA
SCHEMBL1662848 0.71
Hydrochloric Acid SCHEMBL28139054 0.70
SCHEMBL7841684 0.70 DHFR (0.38) PARP1MAPTNPC1RAB9AKMT2A
SCHEMBL7852167 0.70 DHFR (0.38) PARP1MAPTNPC1RAB9AMEN1
SCHEMBL6151295 0.68 PARP1 (0.47) BCAT2PARP1MAPTNPC1LMNA
SCHEMBL25298549 0.67 MYC (0.39) BCAT2MAPTNPC1RAB9ALMNA
SCHEMBL1254367 0.67 BRD4 (0.47) PTGS1PDCD1CD274MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105283451-B Novel inhibitors of viral replication 鲁汶天主教大学 2021-01-26 CN disclosed
CN-105283451-A Novel viral replication inhibitors UNIV LEUVEN KATH 2016-01-27 CN disclosed