SCHEMBL6151295

SCHEMBL6151295

NC(=O)n1ccc(-c2ccccc2)c1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.47
BCAT2 O15382 2/20 0.44
LMNA P02545 1/20 0.37
MAPT P10636 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
GAA P10253 1/20 0.37
PABPC1 P11940 1/20 0.37
KMT2A Q03164 1/20 0.37
BACE1 P56817 2/20 0.36
CTSD P07339 1/20 0.36
SCN9A Q15858 1/20 0.36
FGFR1 P11362 1/20 0.35
SRC P12931 1/20 0.35
FGFR2 P21802 1/20 0.35
FGFR4 P22455 1/20 0.35
FGFR3 P22607 1/20 0.35
CRHBP P24387 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29395257 0.80 PARP1 (0.46) PARP1BCAT2LMNAMAPTTDP1
SCHEMBL27645536 0.76 BCAT2 (0.43) PARP1BCAT2LMNAMAPTTDP1
SCHEMBL15380745 0.69 PARP1 (0.46) PARP1BCAT2LMNAMAPTTDP1
Carbamic Acid SCHEMBL29581535 0.68 BCAT2 (0.67) PARP1BCAT2LMNAMAPTTDP1
Carbamic Acid SCHEMBL27551243 0.68 BCAT2 (0.67) PARP1BCAT2LMNAMAPTTDP1
Urea SCHEMBL1953346 0.68 BCAT2 (0.67) PARP1BCAT2LMNAMAPTTDP1
SCHEMBL28045914 0.68 BCAT2 (0.42) PARP1BCAT2LMNAMAPTKDM4E
SCHEMBL9458564 0.66 ALDH1A1 (0.49) LMNAKDM4ENPC1KMT2ABACE1
SCHEMBL28856325 0.66 BACE1 (0.36) MAPTKDM4ENPC1BACE1HSD17B10
SCHEMBL6842022 0.66 BCAT2 (0.63) PARP1BCAT2LMNAMAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1753668-A 1, 5-diaryl pyrrole-3-carboxamide derivatives and their use as cannabinoid receptor modulators ASTRAZENECA AB (SE) 2006-03-29 CN claimed
CN-113943242-B Preparation method of polysubstituted pyrrole compound 浙江工业大学 2023-08-15 CN disclosed
CN-113943242-A Preparation method of polysubstituted pyrrole compound 浙江工业大学 2022-01-18 CN disclosed
CN-1753668-A 1, 5-diaryl pyrrole-3-carboxamide derivatives and their use as cannabinoid receptor modulators ASTRAZENECA AB (SE) 2006-03-29 CN disclosed
EP-1592404-A1 AQUEOUS DISPERSION COMPRISING STABLE NANOPARTICLES OF A WATER-INSOLUBLE PYRROLE CARBOXAMIDE AND AN EXCIPIENT LIKE MIDDLE CHAIN TRIGLYCERIDES AstraZeneca AB (SE) 2005-11-09 EP disclosed
WO-2004069227-A1 AQUEOUS DISPERSION COMPRISING STABLE NANOPARTICLES OF A WATER-INSOLUBLE PYRROLE CARBOXAMIDE AND EXCIPIENT LIKE MIDDLE CHAIN TRIGLYCERIDES ASTRAZENECA AB (SE) 2004-08-19 WO disclosed