SCHEMBL28046049

SCHEMBL28046049

O=C(C(CBr)c1cccc([N+](=O)[O-])c1F)C(CBr)c1cccc([N+](=O)[O-])c1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.44
TSHR P16473 2/20 0.44
GPR35 Q9HC97 2/20 0.40
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.37
TDP1 Q9NUW8 5/20 0.37
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
CTSD P07339 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MAPT P10636 2/20 0.35
MAPK1 P28482 1/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
GLA P06280 1/20 0.35
POLB P06746 1/20 0.35
RECQL P46063 1/20 0.35
APEX1 P27695 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27437418 0.84 CYP1A2 (0.60) CYP1A2TSHRGPR35ALDH1A1MEN1
SCHEMBL28159152 0.78 CES2 (0.47) MEN1KMT2A
SCHEMBL28046050 0.77 CYP1A2 (0.37) CYP1A2TSHRGPR35ALDH1A1SMN1; SMN2
SCHEMBL16119496 0.76 CYP1A2 (0.47) CYP1A2TSHRGPR35ALDH1A1SMN1; SMN2
SCHEMBL29509474 0.74 TDP1 (0.47) CYP1A2TSHRGPR35ALDH1A1SMN1; SMN2
SCHEMBL16797211 0.74 TDP1 (0.47) CYP1A2TSHRGPR35ALDH1A1SMN1; SMN2
SCHEMBL18867119 0.74 TDP1 (0.47) CYP1A2TSHRGPR35ALDH1A1SMN1; SMN2
SCHEMBL22499481 0.74 GPR35 (0.43) CYP1A2TSHRGPR35ALDH1A1SMN1; SMN2
SCHEMBL10776693 0.73 ALDH1A1 (0.49) TSHRALDH1A1SMN1; SMN2TDP1MEN1
SCHEMBL27841207 0.73 TDP1 (0.46) CYP1A2TSHRGPR35ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105228983-A The compound regulated for kinases and indication thereof PLEXXIKON INC 2016-01-06 CN disclosed