SCHEMBL28046252

SCHEMBL28046252

Nc1cccc(Cc2ccccc2F)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 2/20 0.46
MPO P05164 1/20 0.46
ALDH1A1 P00352 4/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
NPC1 O15118 1/20 0.43
HTT P42858 1/20 0.43
RAB9A P51151 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
TAAR1 Q96RJ0 1/20 0.42
TLR8 Q9NR97 1/20 0.42
TLR7 Q9NYK1 1/20 0.42
APP P05067 1/20 0.41
BACE1 P56817 1/20 0.41
IDO1 P14902 2/20 0.40
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
PTGER1 P34995 2/20 0.40
KCNH3 Q9ULD8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28043564 0.81 MPO (0.48) MPOAPPBACE1NOS3NOS1
SCHEMBL4721 0.79 ADORA2A (0.41) ADORA2AMPOALDH1A1L3MBTL1NPC1
SCHEMBL9391654 0.79 LTA4H (0.44) MPOALDH1A1TAAR1TLR8TLR7
SCHEMBL10573978 0.78 MPO (0.51) ADORA2AMPOALDH1A1L3MBTL1NPC1
SCHEMBL29758354 0.73 BACE1 (0.50) ADORA2AALDH1A1L3MBTL1TLR8APP
SCHEMBL1402167 0.73 BACE1 (0.50) ADORA2AALDH1A1L3MBTL1TLR8APP
SCHEMBL9395340 0.73 KCNH3 (0.47) ADORA2AMPOL3MBTL1RAB9ATAAR1
SCHEMBL28824419 0.72 ADORA2A (0.47) ADORA2AMPOAPPBACE1NOS3
SCHEMBL9953712 0.72 L3MBTL1 (0.50) ALDH1A1L3MBTL1NPC1HTTRAB9A
SCHEMBL3301625 0.71 TAAR1 (0.59) MPOALDH1A1L3MBTL1TAAR1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105324380-A Pyrrolo[2,3-b]pyridine cdk9 kinase inhibitors ABBVIE INC 2016-02-10 CN disclosed