SCHEMBL28047884

SCHEMBL28047884

COC(=O)NC1CCCC(CN)C1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.42
EPHX1 P07099 6/20 0.39
NPSR1 Q6W5P4 1/20 0.38
CYP2D6 P10635 1/20 0.37
SMYD3 Q9H7B4 4/20 0.36
HPGD P15428 2/20 0.36
KMT2A Q03164 1/20 0.36
EPHX2 P34913 1/20 0.35
CCR3 P51677 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25525583 0.84 BTK (0.62) BTKEPHX1KMT2A
SCHEMBL6643733 0.84 BTK (0.62) BTKEPHX1KMT2A
SCHEMBL7958929 0.82 BTK (0.44) BTKEPHX1NPSR1HPGDKMT2A
SCHEMBL8162383 0.82 EPHX1 (0.44) BTKEPHX1NPSR1HPGDKMT2A
SCHEMBL7790384 0.82 BTK (0.51) BTKEPHX1NPSR1CYP2D6KMT2A
SCHEMBL16513497 0.81 CYP2D6 (0.47) BTKEPHX1CYP2D6SMYD3HPGD
SCHEMBL12500923 0.81 ALDH1A1 (0.43) BTKEPHX1NPSR1HPGDKMT2A
SCHEMBL8163075 0.79 EPHX1 (0.47) BTKEPHX1NPSR1HPGDKMT2A
SCHEMBL423315 0.78
SCHEMBL10007376 0.77 BTK (0.45) BTKEPHX1NPSR1CYP2D6KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105189481-A Pyridine cdk9 kinase inhibitors ABBVIE INC 2015-12-23 CN disclosed