SCHEMBL28048054

SCHEMBL28048054

CCCCc1c(C(F)(F)F)c(-c2ccccc2)nc2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 2/20 0.48
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
HPGD P15428 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
TSHR P16473 1/20 0.47
HSD17B10 Q99714 1/20 0.47
TLR8 Q9NR97 5/20 0.45
BCHE P06276 1/20 0.44
ACHE P22303 1/20 0.44
ADORA3 P0DMS8 2/20 0.44
NUDT1 P36639 1/20 0.43
ADORA1 P30542 1/20 0.42
PARP1 P09874 1/20 0.42
PDE10A Q9Y233 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3731476 0.77 KDM4E (0.78) KDM4EALDH1A1GAAHPGDCYP1A2
SCHEMBL27931300 0.76 ADORA2A (0.56) TACR3KDM4EALDH1A1GAAHPGD
SCHEMBL28160159 0.74 TACR3 (0.54) TACR3KDM4EALDH1A1GAAHPGD
SCHEMBL28048083 0.74 LMNA (0.49) KDM4EALDH1A1GAAHPGDCYP1A2
SCHEMBL27832687 0.74 KDM4E (0.58) KDM4EALDH1A1GAAHPGDCYP1A2
SCHEMBL29114095 0.73 GPR84 (0.38) KDM4EALDH1A1TSHRADORA3
SCHEMBL13972063 0.73 TACR3 (0.64) TACR3ALDH1A1CYP1A2CYP3A4TSHR
SCHEMBL5318703 0.72 KDM4E (0.75) KDM4EALDH1A1GAAHPGDCYP1A2
SCHEMBL28002147 0.72 KDM4E (0.53) TACR3KDM4EALDH1A1GAAHPGD
SCHEMBL30948991 0.71 TLR8 (0.60) KDM4EALDH1A1GAAHPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105175327-A Synthesis method of quinoline derivatives UNIV NANYANG NORMAL 2015-12-23 CN disclosed