SCHEMBL28049121

SCHEMBL28049121

O=S(=O)(c1ccccc1)c1c[nH]c2ncncc12

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 3/20 0.65
PIK3C3 Q8NEB9 1/20 0.47
HTR6 P50406 6/20 0.43
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
SLC6A2 P23975 2/20 0.39
FFAR2 O15552 1/20 0.39
HTR2A P28223 1/20 0.38
CCNE2 O96020 1/20 0.38
CCNE1 P24864 1/20 0.38
CDK2 P24941 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28081600 0.86 MAPT (0.49) METPIK3C3
SCHEMBL28074661 0.83 MET (0.46) METPIK3C3SLC6A2NAMPT
SCHEMBL3889418 0.79 MET (1.00) METPIK3C3HTR6
SCHEMBL16913783 0.77 MET (0.62) METPIK3C3HTR6HDAC3HDAC4
SCHEMBL28128723 0.77 MET (0.47) METHTR6HDAC3HDAC4HDAC1
SCHEMBL1093217 0.76 RPS6KA5 (0.40) MET
SCHEMBL3890925 0.75 MET (0.58) METPIK3C3HTR6HDAC3HDAC4
SCHEMBL28049211 0.73 MET (0.54) METPIK3C3HTR6SLC6A2FFAR2
SCHEMBL28128689 0.72 FFAR2 (0.56) METPIK3C3HTR6HDAC3HDAC4
SCHEMBL4494776 0.70 HTR6 (0.58) METPIK3C3HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102665718-B Heterocyclic compounds useful as PDK1 inhibitors MILLENNIUM PHARMACEUTICALS, INC. (US) 2016-03-09 CN disclosed