SCHEMBL28049476

SCHEMBL28049476

CC[CH]C(CCC(C)C)c1cccc(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.43
DAO P14920 1/20 0.42
HTR2A P28223 2/20 0.41
HTR2B P41595 2/20 0.41
HTR2C P28335 1/20 0.41
MC4R P32245 1/20 0.41
SLC6A4 P31645 3/20 0.40
SIGMAR1 Q99720 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
ADRA2C P18825 1/20 0.40
ADRA1A P35348 1/20 0.40
DRD3 P35462 1/20 0.40
OPRK1 P41145 1/20 0.40
SLC6A2 P23975 2/20 0.39
IDO1 P14902 1/20 0.38
TDO2 P48775 1/20 0.38
ACP3 P15309 2/20 0.38
CES2 O00748 1/20 0.38
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28049523 0.85 PNMT (0.45) PNMTDAOHTR2AHTR2BHTR2C
SCHEMBL28049473 0.84 PNMT (0.42) PNMTDAOHTR2AHTR2BHTR2C
SCHEMBL28049563 0.77 ACP3 (0.42) PNMTDAOHTR2AHTR2BHTR2C
SCHEMBL7929105 0.72 PNMT (0.50) PNMTDAOHTR2AHTR2BHTR2C
SCHEMBL24779791 0.72 PNMT (0.53) PNMTDAOHTR2AHTR2BHTR2C
SCHEMBL10274869 0.72 PNMT (0.53) PNMTDAOHTR2AHTR2BHTR2C
SCHEMBL25894263 0.72 PNMT (0.53) PNMTDAOHTR2AHTR2BHTR2C
SCHEMBL28032115 0.71 EPHX1 (0.48) PNMTDAOMC4RIDO1TDO2
SCHEMBL7533204 0.71 PNMT (0.49) PNMTHTR2AHTR2BHTR2CMC4R
SCHEMBL255035 0.70 PNMT (0.55) PNMTDAOHTR2AHTR2BHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102369188-B As the replacement niacinamide of KCNQ2/3 conditioning agent GRUNENTHAL GMBH (DE) 2016-03-02 CN claimed
CN-102369188-B As the replacement niacinamide of KCNQ2/3 conditioning agent GRUNENTHAL GMBH (DE) 2016-03-02 CN disclosed