SCHEMBL28049563

SCHEMBL28049563

CC[CH]C(Cc1ccc(F)cc1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACP3 P15309 2/20 0.42
HTR2A P28223 2/20 0.41
HTR2B P41595 2/20 0.41
HTR2C P28335 1/20 0.41
PNMT P11086 1/20 0.40
LMNA P02545 3/20 0.40
SIGMAR1 Q99720 1/20 0.40
MAPT P10636 1/20 0.40
ADRA2C P18825 1/20 0.40
SLC6A4 P31645 1/20 0.40
ADRA1A P35348 1/20 0.40
DRD3 P35462 1/20 0.40
OPRK1 P41145 1/20 0.40
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39
OPRL1 P41146 1/20 0.39
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28049466 0.86 ACP3 (0.46) ACP3HTR2AHTR2BHTR2CPNMT
SCHEMBL28049476 0.77 PNMT (0.43) ACP3HTR2AHTR2BHTR2CPNMT
SCHEMBL28049473 0.76 PNMT (0.42) ACP3HTR2AHTR2BHTR2CPNMT
SCHEMBL27689629 0.69 ACP3 (0.46) ACP3HTR2AHTR2BHTR2CPNMT
SCHEMBL11217606 0.69 NFE2L2 (0.34) LMNAMAPTMEN1KMT2AKCNH2
SCHEMBL20762538 0.68 ACP3 (0.57) ACP3HTR2AHTR2BHTR2CPNMT
SCHEMBL20350341 0.68 HTR2A (0.50) ACP3HTR2AHTR2BHTR2CPNMT
SCHEMBL7533204 0.68 PNMT (0.49) ACP3HTR2AHTR2BHTR2CPNMT
SCHEMBL27516633 0.67 CNR2 (0.38) SLC6A9IDO1TDO2
SCHEMBL19593126 0.67 PNMT (0.54) ACP3HTR2AHTR2BHTR2CPNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102369188-B As the replacement niacinamide of KCNQ2/3 conditioning agent GRUNENTHAL GMBH (DE) 2016-03-02 CN claimed
CN-102369188-B As the replacement niacinamide of KCNQ2/3 conditioning agent GRUNENTHAL GMBH (DE) 2016-03-02 CN disclosed