SCHEMBL28049578

SCHEMBL28049578

C[CH]C(Cc1ccc(F)c(F)c1)c1ccc(F)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 2/20 0.37
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
TRPA1 O75762 1/20 0.34
HTT P42858 3/20 0.33
ALDH1A1 P00352 1/20 0.33
MAOB P27338 1/20 0.33
TAAR1 Q96RJ0 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
DPP4 P27487 3/20 0.32
MITF O75030 1/20 0.32
LMNA P02545 1/20 0.32
CNR1 P21554 1/20 0.32
CNR2 P34972 1/20 0.32
GPR35 Q9HC97 1/20 0.32
GPR55 Q9Y2T6 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28049484 0.86 TRPA1 (0.44) PTPN1TRPA1HTTALDH1A1MAOB
SCHEMBL28049460 0.81 TAAR1 (0.40) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL28049485 0.72 ALDH1A1 (0.44) CYP3A4CYP2D6HTTALDH1A1TAAR1
SCHEMBL6005258 0.70 PTPN1 (0.49) PTPN1DPP4PTGDR2
SCHEMBL28015442 0.70 TRPA1 (0.41) TRPA1HTT
SCHEMBL2623873 0.69 GABRA1 (0.48) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL9176216 0.69 GABRA1 (0.48) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL28049466 0.69 ACP3 (0.46) CYP1A2CYP3A4CYP2D6CYP2C19ALDH1A1
SCHEMBL23231694 0.67 HTT (0.42) HTTALDH1A1MAOBDPP4DPP8
SCHEMBL14478273 0.66 SLC6A2 (0.55) TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102369188-B As the replacement niacinamide of KCNQ2/3 conditioning agent GRUNENTHAL GMBH (DE) 2016-03-02 CN claimed
CN-102369188-B As the replacement niacinamide of KCNQ2/3 conditioning agent GRUNENTHAL GMBH (DE) 2016-03-02 CN disclosed