SCHEMBL28051435

SCHEMBL28051435

FC(F)(F)c1ccc(Nc2ncnc(Nc3cccc(Cl)c3)n2)cc1

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.56
APP P05067 3/20 0.54
IDH2 P48735 2/20 0.54
SYK P43405 1/20 0.51
CTSC P53634 4/20 0.51
FADS1 O60427 1/20 0.51
TNNI3K Q59H18 1/20 0.50
AURKA O14965 2/20 0.48
CDC7 O00311 1/20 0.48
CDK1 P06493 2/20 0.47
KCNH3 Q9ULD8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28051330 0.86 ADORA3 (0.59) KDM4EAPPSYKTNNI3KKCNH3
SCHEMBL3206970 0.85 AURKA (0.70) SYKAURKACDK1
SCHEMBL28037898 0.84 KCNH2 (0.54) KDM4EIDH2SYKCDK1KCNH3
Trifluoromethylbenzene SCHEMBL28051437 0.84 KDM4E (0.75) KDM4EIDH2SYKCTSCAURKA
SCHEMBL6033558 0.80 APP (0.48) KDM4EAPPSYKCTSCKCNH3
SCHEMBL28051328 0.78 TRPV1 (0.58) KDM4ECTSCAURKACDC7CDK1
SCHEMBL4947229 0.78 SYK (0.56) SYKFADS1TNNI3KCDK1
SCHEMBL6583848 0.77 CAMK2D (0.64) SYKFADS1CDK1
SCHEMBL2946515 0.77 PLK1 (0.77) SYK
SCHEMBL28051498 0.77 IDH2 (0.53) KDM4EIDH2SYKTNNI3KCDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105294588-A Fluorotriazine-containing derivative, and preparation method and use thereof WUHAN INST TECHNOLOGY 2016-02-03 CN disclosed