SCHEMBL28051328

SCHEMBL28051328

FC(F)(F)c1ccc(Nc2ncnc(Nc3ccccc3Cl)n2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 3/20 0.58
PTK2 Q05397 1/20 0.53
NPC1 O15118 1/20 0.51
RAB9A P51151 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
AURKA O14965 6/20 0.49
AURKB Q96GD4 4/20 0.47
JAK2 O60674 2/20 0.47
MAPK8 P45983 1/20 0.47
CDK2 P24941 2/20 0.47
CDC7 O00311 1/20 0.47
DAPK3 O43293 1/20 0.47
PAK4 O96013 1/20 0.47
PIM1 P11309 1/20 0.47
FLT3 P36888 1/20 0.47
GSK3B P49841 1/20 0.47
CDK9 P50750 1/20 0.47
CDK5 Q00535 1/20 0.47
DYRK1A Q13627 1/20 0.47
MELK Q14680 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28037898 0.84 KCNH2 (0.54) PTK2RAB9ASMN1; SMN2JAK2MAPK8
SCHEMBL14214726 0.84 KDM4E (0.50) TRPV1PTK2RAB9ASMN1; SMN2JAK2
SCHEMBL28051330 0.83 ADORA3 (0.59) TRPV1SMN1; SMN2CDK2STK17AKCNH3
SCHEMBL4584219 0.82 TRPV1 (0.54) TRPV1PTK2NPC1RAB9ASMN1; SMN2
Trifluoromethylbenzene SCHEMBL28051329 0.82 LMNA (0.61) TRPV1NPC1RAB9ASMN1; SMN2AURKA
SCHEMBL6033558 0.80 APP (0.48) TRPV1SMN1; SMN2CDK2KCNH3CTSC
SCHEMBL28051435 0.78 KDM4E (0.56) AURKACDC7KCNH3CTSCCDK1
SCHEMBL28051498 0.77 IDH2 (0.53) PTK2RAB9ASMN1; SMN2JAK2CDK2
SCHEMBL13801564 0.75 TRPV1 (0.66) TRPV1
SCHEMBL18434160 0.75 HDAC3 (0.54) TRPV1PTK2NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105294588-A Fluorotriazine-containing derivative, and preparation method and use thereof WUHAN INST TECHNOLOGY 2016-02-03 CN disclosed