SCHEMBL28052129

SCHEMBL28052129

CN(Cc1ccccc1)CC1CC(=O)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.45
JAK1 P23458 1/20 0.45
NR1H2 P55055 2/20 0.41
NR1H3 Q13133 2/20 0.41
GHSR Q92847 6/20 0.41
PARP1 P09874 1/20 0.41
ATM Q13315 2/20 0.39
HCRTR1 O43613 1/20 0.39
STS P08842 1/20 0.39
KDM1A O60341 1/20 0.38
AKT1 P31749 1/20 0.38
HSD11B1 P28845 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL582271 0.84 NR1H2 (0.53) JAK2JAK1NR1H2NR1H3PARP1
SCHEMBL15353299 0.84 NR1H2 (0.53) JAK2JAK1NR1H2NR1H3PARP1
SCHEMBL15880038 0.84 NR1H2 (0.53) JAK2JAK1NR1H2NR1H3PARP1
SCHEMBL7520525 0.76 ABCB1 (0.49) GHSRPARP1
SCHEMBL31122968 0.75 PARP1 (0.39) NR1H2NR1H3PARP1ATMKDM1A
SCHEMBL19389933 0.75 GPR119 (0.43) JAK2JAK1NR1H2NR1H3GHSR
SCHEMBL3941124 0.74 ATM (0.43) PARP1ATMKDM1A
SCHEMBL21360450 0.74 ATM (0.43) PARP1ATMKDM1A
SCHEMBL19390116 0.74 ATM (0.41) NR1H2PARP1ATMKDM1A
SCHEMBL5838439 0.74 ALDH1A1 (0.40) NR1H2NR1H3ATMKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105646332-B Aminomethylpiperidine analog derivative and preparation method thereof and medicinal usage 复旦大学 2018-05-25 CN disclosed
CN-105646332-A Aminomethylpiperidine derivatives, and preparation method and pharmaceutical application thereof 复旦大学 2016-06-08 CN disclosed