SCHEMBL28052878

SCHEMBL28052878

COC(=O)c1cncc(CN2CCN(OC(=O)C(C)(C)C)CC2)c1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 3/20 0.44
ATM Q13315 1/20 0.41
KDM1A O60341 2/20 0.40
FAAH O00519 2/20 0.39
KLKB1 P03952 3/20 0.39
KLK1 P06870 3/20 0.39
CHKA P35790 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 2/20 0.38
GAA P10253 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HSD17B10 Q99714 1/20 0.38
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28052661 0.83 MEN1 (0.53) FAAHSMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL28272975 0.82 CHKA (0.56) ATMCHKASMN1; SMN2ALDH1A1GAA
SCHEMBL29390664 0.82 ACKR3 (0.46) ACKR3ATMKDM1AFAAHALDH1A1
SCHEMBL16486773 0.82 ACKR3 (0.46) ACKR3ATMKDM1AFAAHALDH1A1
SCHEMBL28289204 0.80 KDM4E (0.34) ATMALDH1A1MEN1KMT2A
SCHEMBL23013506 0.80 ALDH1A1 (0.57) ACKR3FAAHKLKB1KLK1SMN1; SMN2
SCHEMBL16486820 0.80 FAAH (0.47) ACKR3ATMKDM1AFAAHCHKA
SCHEMBL28248650 0.80 KLKB1 (0.46) ACKR3ATMKDM1AFAAHKLKB1
SCHEMBL16486396 0.78 CHRM3 (0.50) ACKR3ATMFAAHKLKB1KLK1
SCHEMBL27844847 0.76 CHRNB2 (0.54) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105683179-A Inhibitors of plasma kallikrein 卡尔维斯塔制药有限公司 2016-06-15 CN disclosed