SCHEMBL28053342

SCHEMBL28053342

NS(=O)(=O)c1cc(-c2cc(Cl)cnc2O)sc1-c1cc(Cl)cnc1O

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
ALOX5AP P20292 1/20 0.31
FEN1 P39748 1/20 0.31
S100A9 P06702 1/20 0.31
PLAU P00749 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28053246 0.77 GCK (0.34) CA1CA2ALOX5APFEN1PLAU
SCHEMBL28053345 0.68 APLNR (0.50) PTGS1PTGS2CA1CA2S100A9
SCHEMBL28053340 0.63 PTGS1 (0.42) PTGS1PTGS2CA1CA2S100A9
SCHEMBL6619882 0.62 CA1 (0.44) PTGS1PTGS2CA1CA2
SCHEMBL21931144 0.62 LMNA (0.38) CA1CA2S100A9PLAU
SCHEMBL10178016 0.61 CA1 (0.43) PTGS1PTGS2CA1CA2
SCHEMBL31028780 0.61 CA1 (0.43) PTGS1PTGS2CA1CA2ALOX5AP
SCHEMBL454507 0.60
SCHEMBL6069906 0.60 PTGS2 (0.63) PTGS1PTGS2
SCHEMBL16235676 0.59 S100A9 (0.55) S100A9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105377837-A N-(heteroaryl)-sulfonamide derivatives useful as S100-inhibitors ACTIVE BIOTECH AB 2016-03-02 CN claimed
CN-105377837-A N-(heteroaryl)-sulfonamide derivatives useful as S100-inhibitors ACTIVE BIOTECH AB 2016-03-02 CN disclosed