SCHEMBL28053345

SCHEMBL28053345

NS(=O)(=O)c1cncc(-c2cc(Cl)cnc2O)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.50
PTGS2 P35354 8/20 0.43
PTGS1 P23219 6/20 0.43
S100A9 P06702 1/20 0.41
PIK3CG P48736 3/20 0.40
PIK3CD O00329 2/20 0.40
SCN10A Q9Y5Y9 1/20 0.40
PTGES2 Q9H7Z7 1/20 0.37
CA1 P00915 3/20 0.35
CA2 P00918 3/20 0.35
CA9 Q16790 3/20 0.35
CA12 O43570 2/20 0.35
MKNK1 Q9BUB5 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
CDK2 P24941 1/20 0.34
PIK3CA P42336 1/20 0.34
CA4 P22748 2/20 0.33
CA5A P35218 2/20 0.33
CA5B Q9Y2D0 2/20 0.33
ABCC4 O15439 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28053322 0.78 APLNR (0.51) APLNRPTGS2PTGS1PIK3CGPIK3CD
SCHEMBL1775244 0.75 APLNR (0.59) APLNRPTGS2PTGS1S100A9PIK3CG
SCHEMBL28053340 0.74 PTGS1 (0.42) APLNRPTGS2PTGS1S100A9PTGES2
SCHEMBL6069906 0.72 PTGS2 (0.63) PTGS2PTGS1ABCC4ABCB11PDE4D
SCHEMBL28053243 0.71 APLNR (0.47) APLNRPTGS2PIK3CGPIK3CDSCN10A
SCHEMBL6069927 0.71 PTGS2 (0.49) PTGS2PTGS1ABCC4ABCB11PDE4D
SCHEMBL5989061 0.70 CYP2A6 (0.50) PTGS2PTGS1
SCHEMBL11690551 0.69 APLNR (0.71) APLNRPIK3CGPIK3CDCA1CA2
SCHEMBL18247080 0.68 APLNR (1.00) APLNRPTGS2PTGS1PIK3CGPIK3CD
SCHEMBL28053342 0.68 PTGS1 (0.36) PTGS2PTGS1S100A9CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105377837-A N-(heteroaryl)-sulfonamide derivatives useful as S100-inhibitors ACTIVE BIOTECH AB 2016-03-02 CN claimed
CN-105377837-A N-(heteroaryl)-sulfonamide derivatives useful as S100-inhibitors ACTIVE BIOTECH AB 2016-03-02 CN disclosed