SCHEMBL28053546

SCHEMBL28053546

NCc1cccc(C2CCCN(C(=O)c3ccccn3)C2)c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
PDE2A O00408 1/20 0.50
SCD5 Q86SK9 2/20 0.48
ALDH1A1 P00352 1/20 0.47
F10 P00742 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
PLA2G1B P04054 1/20 0.47
ATG4B Q9Y4P1 1/20 0.47
PROKR1 Q8TCW9 2/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
SCD O00767 1/20 0.46
EPHX2 P34913 1/20 0.46
TPSAB1 Q15661 1/20 0.46
CSF1R P07333 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16446230 0.84 PROKR1 (0.64) MEN1KMT2APDE2ASCD5L3MBTL1
SCHEMBL28853754 0.81 DRD3 (0.50) ALDH1A1TPSAB1
SCHEMBL28189351 0.80 PROKR1 (0.50) ALDH1A1PROKR1CYP3A4TPSAB1
SCHEMBL28053449 0.79 PROKR1 (0.75) PROKR1
Ammonia Solution, Strong SCHEMBL28053450 0.79 PROKR1 (0.49) ALDH1A1PROKR1CYP3A4TPSAB1
SCHEMBL28189333 0.78 BTK (0.44) ALDH1A1F10
SCHEMBL4036337 0.76 BCL9 (0.61) MEN1KMT2APROKR1
SCHEMBL28853756 0.74 DRD2 (0.48) TPSAB1
SCHEMBL13570456 0.73 F10 (0.45) F10CYP3A4TPSAB1
SCHEMBL8350555 0.73 SCD5 (0.53) MEN1KMT2APDE2ASCD5L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105452233-A Piperidine and azepane derivatives as prokineticin receptor modulators TAKEDA PHARMACEUTICALS CO 2016-03-30 CN claimed
CN-105452233-A Piperidine and azepane derivatives as prokineticin receptor modulators TAKEDA PHARMACEUTICALS CO 2016-03-30 CN disclosed