SCHEMBL28056097

SCHEMBL28056097

O=C(O)c1ccc(CCc2ccc(Cl)cc2)c(C(=O)O)c1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
TSHR P16473 2/20 0.48
ALOX15 P16050 1/20 0.48
LMNA P02545 2/20 0.48
DAO P14920 1/20 0.48
MAPT P10636 2/20 0.46
NR4A2 P43354 2/20 0.45
AKR1C3 P42330 1/20 0.45
MRGPRX4 Q96LA9 1/20 0.45
SRD5A2 P31213 1/20 0.44
CTRC Q99895 1/20 0.43
NR4A1 P22736 1/20 0.42
EBP Q15125 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28052169 0.88 TSHR (0.44) ALDH1A1TSHRLMNA
SCHEMBL27383637 0.85 TSHR (0.51) ALDH1A1TSHRDAOMAPT
SCHEMBL28052882 0.84 CES2 (0.45) ALDH1A1TSHR
SCHEMBL12063879 0.84 KDM5A (0.46) TSHRNR4A2
SCHEMBL27734240 0.84 TSHR (0.44) ALDH1A1TSHRALOX15MAPTMEN1
SCHEMBL28855166 0.84 NR4A2 (0.55) ALDH1A1TSHRNR4A2MRGPRX4SRD5A2
SCHEMBL11687234 0.84 RXRA (0.45) TSHRAKR1C3MRGPRX4SRD5A2MEN1
SCHEMBL23040963 0.84 RXRA (0.51) ALDH1A1NR4A2AKR1C3MRGPRX4MEN1
SCHEMBL28119542 0.83 ALDH1A1 (0.50) ALDH1A1TSHRALOX15MAPTNR4A2
SCHEMBL6387117 0.82 ALDH1A1 (0.67) ALDH1A1TSHRLMNADAOMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105407888-A Novel bicyclic bromodomain inhibitors ZENITH EPIGENETICS CORP 2016-03-16 CN claimed
CN-105407888-A Novel bicyclic bromodomain inhibitors ZENITH EPIGENETICS CORP 2016-03-16 CN disclosed