SCHEMBL28056834

SCHEMBL28056834

CC(C)(C)OC(=O)NCC(=O)NS(=O)(=O)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.49
CA12 O43570 2/20 0.49
CA7 P43166 1/20 0.49
CA14 Q9ULX7 1/20 0.49
EGFR P00533 4/20 0.48
ERBB2 P04626 4/20 0.48
BCL2 P10415 1/20 0.46
KDM4E B2RXH2 1/20 0.44
CA2 P00918 3/20 0.44
NPFFR1 Q9GZQ6 1/20 0.43
NPFFR2 Q9Y5X5 1/20 0.43
PPARA Q07869 1/20 0.43
ACACB O00763 1/20 0.43
CA9 Q16790 1/20 0.42
EPHX2 P34913 1/20 0.42
SIGMAR1 Q99720 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20153436 0.88 MEP1B (0.47) CA1CA12CA7CA14CA2
SCHEMBL1161283 0.86 CA1 (0.50) CA1CA12CA7CA14EGFR
SCHEMBL3929114 0.85 EGFR (0.53) CA1CA12EGFRERBB2CA2
SCHEMBL5394506 0.84 CA1 (0.57) CA1CA12CA7CA14EGFR
SCHEMBL28254302 0.83 EGFR (0.51) CA1EGFRERBB2KDM4ECA2
SCHEMBL8493222 0.80 MMP2 (0.48)
SCHEMBL21780201 0.80 MALT1 (0.47) CA1CA12CA7CA14BCL2
SCHEMBL8493227 0.80 CTSS (0.41) CA1CA12CA7CA14BCL2
SCHEMBL3368185 0.80 CA12 (0.57) CA1CA12CA7CA2CA9
SCHEMBL5071878 0.79 PTGS2 (0.69) CA1CA12CA7CA14CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109384778-B Use of a compound or a pharmaceutically acceptable salt thereof for the manufacture of a medicament for the treatment of a disease, health condition or disorder 赛克里翁治疗有限公司 2022-12-13 CN disclosed
CN-110016020-B Compound or pharmaceutically acceptable salt thereof, application and pharmaceutical composition thereof 赛克里翁治疗有限公司 2022-07-26 CN disclosed
CN-108912111-B Compounds and pharmaceutical compositions 赛克里翁治疗有限公司 2021-09-14 CN disclosed
CN-110016020-A Compound or pharmaceutically acceptable salt thereof, application and pharmaceutical composition thereof 铁木医药有限公司 2019-07-16 CN disclosed
CN-109384778-A Use of a compound or a pharmaceutically acceptable salt thereof for the manufacture of a medicament for the treatment of a disease, health condition or disorder 铁木医药有限公司 2019-02-26 CN disclosed
CN-109369635-A Compound or pharmaceutically acceptable salt thereof, application and pharmaceutical composition thereof 铁木医药有限公司 2019-02-22 CN disclosed
CN-108912111-A compounds and pharmaceutical compositions 铁木医药有限公司 2018-11-30 CN disclosed
CN-105408328-B sGC stimulators 铁木医药有限公司 2018-11-16 CN disclosed
CN-105408328-A sGC stimulators IRONWOOD PHARMACEUTICALS INC 2016-03-16 CN disclosed