SCHEMBL28056863

SCHEMBL28056863

COC(=O)C1Cc2ccccc2C=N1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 7/20 0.42
MTNR1A P48039 2/20 0.36
MTNR1B P49286 2/20 0.36
POLB P06746 1/20 0.34
GRM7 Q14831 2/20 0.34
CYP1A2 P05177 2/20 0.34
HSD17B10 Q99714 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP2C19 P33261 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16431429 0.80 GAA (0.39) TRPA1GRM7TSHRMEN1KMT2A
SCHEMBL28938653 0.80 FAAH (0.45)
SCHEMBL27453351 0.79 HDAC4 (0.42)
SCHEMBL10658578 0.74 MTNR1A (0.41) MTNR1AMTNR1BPOLBGRM7CYP1A2
SCHEMBL7462076 0.74 TRPA1 (0.38) TRPA1MTNR1AMTNR1BPOLBCYP1A2
SCHEMBL14953404 0.74 KEAP1 (0.35) POLBCYP2C19KMT2A
Hydrochloric Acid SCHEMBL1509729 0.73 KEAP1 (0.35) POLBCYP2C19KMT2A
SCHEMBL28144460 0.73 XIAP (0.40) KMT2A
SCHEMBL28144463 0.73 XIAP (0.40) KMT2A
SCHEMBL23794999 0.72 POLB (0.37) TRPA1MTNR1AMTNR1BPOLBCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105777712-B Tetrahydroisoquinoliderivs derivs and its application 沈阳药科大学 2018-05-22 CN disclosed
CN-105777712-A Tetrahydroisoquinoline derivative and application thereof 沈阳药科大学 2016-07-20 CN disclosed
CN-103732589-B Can be used as the sulphonamide of the replacement of anti-apoptotic BCL inhibitor BRISTOL-MYERS SQUIBB CO. (US) 2016-03-30 CN disclosed