SCHEMBL28058282

SCHEMBL28058282

NC(=O)c1cc(N)cc(F)c1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 5/20 0.43
CES1 P23141 5/20 0.43
DGAT1 O75907 1/20 0.42
MEN1 O00255 5/20 0.37
KMT2A Q03164 5/20 0.37
KDM4E B2RXH2 3/20 0.37
MAPT P10636 3/20 0.37
THRB P10828 3/20 0.37
ALOX15 P16050 2/20 0.37
HSD17B10 Q99714 2/20 0.37
GFER P55789 1/20 0.37
YWHAG P61981 1/20 0.37
HTT P42858 1/20 0.36
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA4 P22748 2/20 0.35
TDP1 Q9NUW8 3/20 0.35
BCHE P06276 1/20 0.34
MAP2K2 P36507 1/20 0.34
MAP2K1 Q02750 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL671650 0.83 KDM4E (0.48) CES2CES1MEN1KMT2AKDM4E
SCHEMBL30739727 0.83 KDM4E (0.48) CES2CES1MEN1KMT2AKDM4E
SCHEMBL477698 0.80 CES2 (0.68) CES2CES1DGAT1CA1CA2
SCHEMBL16006488 0.78 CES2 (0.43) CES2CES1DGAT1KDM4ECA1
SCHEMBL829400 0.77 DGAT1 (0.45) CES2CES1DGAT1CA1CA2
SCHEMBL28085635 0.77 DGAT1 (0.45) CES2CES1DGAT1CA1CA2
SCHEMBL17761393 0.77 MAP2K1 (0.46) CES2CES1DGAT1CA1CA2
SCHEMBL15994788 0.77 DGAT1 (0.60) CES2CES1DGAT1MEN1KMT2A
SCHEMBL15490200 0.75 IKBKB (0.38) DGAT1MEN1KMT2AKDM4EHTT
SCHEMBL4262805 0.75 DGAT1 (0.38) CES2CES1DGAT1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105461585-A 3-aminobenzamide derivative as beta-lactam auxiliary antibiotic, preparation method and application UNIV HONG KONG POLYTECHNIC 2016-04-06 CN disclosed