SCHEMBL28059202

SCHEMBL28059202

Cc1ccnc(C2CNCCO2)n1

nearest known ligand 0.47

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.46
SLC6A3 Q01959 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27635980 0.82 SLC6A3 (0.46) TAAR1SLC6A3
SCHEMBL28071137 0.79
SCHEMBL913262 0.79 DRD2 (0.46)
SCHEMBL28059111 0.78 DRD2 (0.40) TAAR1SLC6A3
SCHEMBL18342698 0.78 SLC6A3 (0.39) TAAR1SLC6A3
Hydrogen Sulfide SCHEMBL28070942 0.77 DRD2 (0.45)
SCHEMBL24001944 0.76 SLC6A3 (0.43) TAAR1SLC6A3
SCHEMBL24009800 0.76 SLC6A3 (0.60) TAAR1SLC6A3
SCHEMBL25170238 0.76 SLC6A3 (0.60) TAAR1SLC6A3
SCHEMBL30403347 0.76 SLC6A3 (0.43) TAAR1SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105814043-B Triazolopyridine derivatives as TNF active regulator UCB生物制药私人有限公司 2019-05-17 CN disclosed
CN-105814049-B Fused tricyclic imdazole derivatives as TNF active regulator UCB生物制药私人有限公司 2019-03-12 CN disclosed
CN-109219608-A FUSED PENTACYCLIC IMIDAZOLE DERIVATIVES AS MODULATORS OF TNF ACTIVITY UCB生物制药私人有限公司 2019-01-15 CN disclosed
CN-109219609-A FUSED HEXACYCLIC IMIDAZOLE DERIVATIVES AS MODULATORS OF TNF ACTIVITY UCB生物制药私人有限公司 2019-01-15 CN disclosed
CN-109195969-A FUSED PENTACYCLIC IMIDAZOLE DERIVATIVES AS MODULATORS OF TNF ACTIVITY UCB生物制药私人有限公司 2019-01-11 CN disclosed
CN-109195968-A FUSED PENTACYCLIC IMIDAZOLE DERIVATIVES AS MODULATORS OF TNF ACTIVITY UCB生物制药私人有限公司 2019-01-11 CN disclosed
CN-105814041-B Benzotriazole derivatives as TNF active regulator UCB生物制药私人有限公司 2018-12-18 CN disclosed
CN-105814065-B Imidazothiazole derivative as TNF active regulator UCB生物制药私人有限公司 2018-11-23 CN disclosed
CN-105814058-B Triazolo-pyridazine derivatives as TNF active regulator UCB生物制药私人有限公司 2018-11-23 CN disclosed
CN-105814047-B Fused tricyclic imdazole derivatives as TNF active regulators UCB生物制药私人有限公司 2018-10-19 CN disclosed
CN-105814059-A Imidazopyrimidine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814051-A Tetrahydroimidazopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814065-A Imidazothiazole derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814050-A Pyrazolopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814025-A Tetrahydrobenzimidazole derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814047-A Fused tricyclic benzimidazoles derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814054-A Fused imidazole and pyrazole derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814049-A Fused tricyclic imidazole derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814043-A Triazolopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
CN-105814045-A Imidazopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed