SCHEMBL28059288

SCHEMBL28059288

CC(C)(C)C1C(Oc2cccc(N)c2)CCN1C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 6/20 0.38
KCNH2 Q12809 3/20 0.38
CHRM3 P20309 6/20 0.37
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
NOTUM Q6P988 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP3A4 P08684 1/20 0.35
POLB P06746 1/20 0.35
CHRM2 P08172 3/20 0.34
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
CPT1A P50416 1/20 0.34
MAOB P27338 1/20 0.34
RIPK1 Q13546 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28826953 0.93 POLB (0.40) OPRK1KCNH2CHRM3CHRNB2CHRNA4
SCHEMBL28059300 0.88 CHRM3 (0.38) OPRK1KCNH2CHRM3CHRNB2CHRNA4
SCHEMBL20658831 0.84 TSHR (0.38) OPRK1KCNH2CHRM3ALDH1A1POLB
SCHEMBL4279118 0.82 CHRM3 (0.36) OPRK1KCNH2CHRM3
SCHEMBL4279130 0.82 CHRM3 (0.36) OPRK1KCNH2CHRM3
SCHEMBL28059315 0.82 SLC6A2 (0.44) CHRNB2CHRNA4ALDH1A1CPT1A
SCHEMBL28053867 0.80 OPRK1 (0.41) OPRK1KCNH2CHRM3POLBCHRM2
SCHEMBL23526972 0.77 EPHX2 (0.42) NOTUMALDH1A1
SCHEMBL23527276 0.75 EPHX2 (0.41) NOTUMALDH1A1
SCHEMBL4102370 0.75 RBP4 (0.38) RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105384695-A Pyrimidine derivative, preparation method therefor and application thereof in medicine SICHUAN HAISCO PHARMACEUTICAL CO LTD 2016-03-09 CN disclosed