SCHEMBL28053867

SCHEMBL28053867

CC(C)(C)C1CC(Oc2cccc(N)c2)CCN1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
OPRK1 P41145 7/20 0.41
KCNH2 Q12809 4/20 0.41
CHRM3 P20309 6/20 0.41
POLB P06746 2/20 0.38
CHRM2 P08172 3/20 0.38
EPHX2 P34913 3/20 0.38
OPRM1 P35372 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28053866 0.84 SLC6A2 (0.50) OPRK1KCNH2CHRM3
SCHEMBL4718944 0.81 HRH1 (0.47) KCNH2
SCHEMBL15639975 0.80 CHRM3 (0.34) OPRK1KCNH2CHRM3POLBEPHX2
SCHEMBL28059288 0.80 OPRK1 (0.38) OPRK1KCNH2CHRM3POLBCHRM2
SCHEMBL8536867 0.80 CCR5 (0.40) CHRM3POLBCHRM2EPHX2
SCHEMBL2196095 0.79 OPRK1 (0.39) OPRK1KCNH2OPRM1
SCHEMBL3985447 0.79 RIPK1 (0.39) OPRM1
SCHEMBL3292130 0.79 OPRK1 (0.49) OPRK1CHRM3EPHX2
SCHEMBL4469103 0.78 HMOX1 (0.36) CHRM3CHRM2EPHX2
SCHEMBL10262344 0.77 KDM1A (0.42) OPRK1KCNH2CHRM3POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105384694-A Substituted aminopyrimidine derivative, preparation method therefor and pharmaceutical application thereof SICHUAN HAISCO PHARMACEUTICAL CO LTD 2016-03-09 CN disclosed
CN-105384695-A Pyrimidine derivative, preparation method therefor and application thereof in medicine SICHUAN HAISCO PHARMACEUTICAL CO LTD 2016-03-09 CN disclosed